SCHEMBL3237174

SCHEMBL3237174

Cc1cnc(NC(=O)CCCCC(C(N)=O)c2ccc(F)cc2N)o1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 17/20 0.41
HDAC3 O15379 17/20 0.41
HDAC2 Q92769 8/20 0.41
NCOR2 Q9Y618 6/20 0.38
HDAC4 P56524 1/20 0.34
MEF2D Q14814 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3237178 0.81 HDAC1 (0.56) HDAC1HDAC3HDAC2NCOR2
SCHEMBL3234097 0.80 HDAC1 (0.48) HDAC1HDAC3HDAC2NCOR2HDAC4
SCHEMBL3228522 0.78 HDAC3 (0.53) HDAC1HDAC3HDAC2HDAC4MEF2D
SCHEMBL3235060 0.78 KDM4E (0.38) HDAC1HDAC3NCOR2NPC1RAB9A
SCHEMBL3238636 0.76 HDAC3 (0.36) HDAC1HDAC3
SCHEMBL3262232 0.76 HDAC1 (0.39) HDAC1HDAC3HDAC2NCOR2
SCHEMBL3227550 0.71 HDAC1 (0.52) HDAC1HDAC3HDAC2NCOR2HDAC4
SCHEMBL3238553 0.71 HDAC1 (0.44) HDAC1HDAC3HDAC2NCOR2MAPT
SCHEMBL3233819 0.70 HDAC3 (0.47) HDAC1HDAC3HDAC2NCOR2HDAC4
SCHEMBL3241863 0.70 HDAC1 (0.52) HDAC1HDAC3HDAC2NCOR2HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO claimed