SCHEMBL3228604

SCHEMBL3228604

COc1ccc([N+](=O)[O-])cn1.COc1ccc2[nH]cc(C=O)c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
PABPC1 P11940 2/20 0.46
ERN1 O75460 2/20 0.43
MAPT P10636 9/20 0.41
HTT P42858 6/20 0.41
LMNA P02545 5/20 0.41
SMN1; SMN2 Q16637 5/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
POLB P06746 1/20 0.41
BLM P54132 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HSPB1 P04792 2/20 0.38
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29953009 0.83 ALDH1A1 (0.49) MEN1KMT2AERN1MAPTALDH1A1
SCHEMBL3035666 0.83 ALDH1A1 (0.49) MEN1KMT2AERN1MAPTALDH1A1
SCHEMBL1851173 0.76 KMT2A (0.70) MEN1KMT2APABPC1ERN1MAPT
SCHEMBL30850667 0.76 KMT2A (0.70) MEN1KMT2APABPC1ERN1MAPT
SCHEMBL23166407 0.73 TXNRD1 (0.47) MAPTHTTMAPK1MTNR1AMTNR1B
SCHEMBL30166982 0.73 TXNRD1 (0.47) MAPTHTTMAPK1MTNR1AMTNR1B
SCHEMBL29954006 0.70 CYP3A4 (0.43) MEN1KMT2AERN1MAPTHTT
SCHEMBL16835850 0.68 KMT2A (0.59) MEN1KMT2APABPC1ERN1MAPT
SCHEMBL18285419 0.66 KMT2A (0.57) MEN1KMT2APABPC1MAPTLMNA
SCHEMBL261553 0.66 MEN1 (0.57) MEN1KMT2APABPC1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010030727-A1 3-SUBSTITUTED-1H-INDOLE, 3-SUBSTITUTED-1H-PYRROLO[2,3-B]PYRIDINE AND 3-SUBSTITUTED-1H-PYRROLO[3,2-B]PYRIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH LLC (US) 2010-03-18 WO disclosed