SCHEMBL3228765

SCHEMBL3228765

CC(CN1CCOCC1)c1ccc(Br)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
KDM4E B2RXH2 3/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
ALOX12 P18054 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
TSHR P16473 2/20 0.50
USP2 O75604 1/20 0.50
HSP90AA1 P07900 1/20 0.49
NTSR1 P30989 1/20 0.49
GFER P55789 1/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
MPI P34949 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11493109 0.95 ALDH1A1 (0.50) ALDH1A1KDM4EL3MBTL1ALOX12NPSR1
SCHEMBL16572388 0.83 ALDH1A1 (0.68) ALDH1A1KDM4EL3MBTL1GFERKMT2A
SCHEMBL5510459 0.83 ALDH1A1 (0.68) ALDH1A1KDM4EL3MBTL1GFERKMT2A
SCHEMBL4060240 0.81 ALDH1A1 (0.47) ALDH1A1KDM4EL3MBTL1ALOX12NPSR1
SCHEMBL11489064 0.81 ALDH1A1 (0.56) ALDH1A1KDM4EL3MBTL1GFERKMT2A
SCHEMBL11493352 0.80 ALDH1A1 (0.46) ALDH1A1TSHRKMT2ALMNAMAPT
SCHEMBL2947238 0.80 TSHR (0.50) ALDH1A1KDM4EL3MBTL1ALOX12NPSR1
SCHEMBL2950084 0.80 KDM4E (0.71) ALDH1A1KDM4EL3MBTL1ALOX12NPSR1
SCHEMBL2947236 0.80 TSHR (0.50) ALDH1A1KDM4EL3MBTL1ALOX12NPSR1
SCHEMBL27775260 0.80 TSHR (0.50) ALDH1A1KDM4EL3MBTL1ALOX12NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010010189-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE AND INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2010-01-28 WO disclosed
WO-2010010184-A1 [1, 2, 4] TRIAZOLO [1, 5-A] PYRIDINES AS JAK INHIBITORS GALAPAGOS NV (BE) 2010-01-28 WO disclosed