SCHEMBL3232171

SCHEMBL3232171

COc1ccc(NC(=O)CCCCCC(=O)Nc2ccc(F)cc2N)c(OC)n1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 17/20 0.55
HDAC3 O15379 13/20 0.55
NCOR2 Q9Y618 1/20 0.53
PIK3CA P42336 5/20 0.45
CDK9 P50750 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3234330 0.93 HDAC1 (0.54) HDAC1HDAC3NCOR2PIK3CACDK9
SCHEMBL3235360 0.85 HDAC3 (0.72) HDAC1HDAC3NCOR2
SCHEMBL7929398 0.82 HDAC1 (0.74) HDAC1HDAC3NCOR2
SCHEMBL7929328 0.82 KCNQ4 (0.43) HDAC1HDAC3NCOR2
SCHEMBL7929314 0.81 HDAC3 (0.52) HDAC1HDAC3
SCHEMBL2618066 0.78 HDAC1 (0.69) HDAC1HDAC3NCOR2
SCHEMBL2618087 0.77 HDAC1 (0.64) HDAC1HDAC3NCOR2
SCHEMBL7931728 0.77 HDAC1 (0.67) HDAC1HDAC3NCOR2
SCHEMBL3234137 0.76 HDAC3 (0.70) HDAC1HDAC3NCOR2
SCHEMBL27757715 0.76 HDAC1 (0.62) HDAC1HDAC3NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO claimed
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed