SCHEMBL3235100

SCHEMBL3235100

Nc1cc(F)ccc1NC(=O)CCCCCC(=O)Nc1nc(CN2CCOCC2)cs1

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 14/20 0.62
HDAC1 Q13547 12/20 0.47
HDAC2 Q92769 4/20 0.46
TNIK Q9UKE5 1/20 0.45
HDAC10 Q969S8 2/20 0.43
NCOR2 Q9Y618 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3262614 0.91 HDAC3 (0.50) HDAC3HDAC1HDAC2HDAC10NCOR2
SCHEMBL3235298 0.83 HDAC1 (0.54) HDAC3HDAC1HDAC2HDAC10NCOR2
SCHEMBL3228076 0.82 HDAC3 (0.55) HDAC3HDAC1HDAC2HDAC10NCOR2
SCHEMBL7933437 0.81 POLB (0.50) HDAC3HDAC1HDAC2HDAC10SMN1; SMN2
SCHEMBL3238457 0.78 HDAC1 (0.56) HDAC3HDAC1HDAC2HDAC10NCOR2
SCHEMBL1937893 0.77 HDAC3 (1.00) HDAC3HDAC1NCOR2
SCHEMBL3237865 0.77 HDAC3 (0.53) HDAC3HDAC1HDAC2HDAC10NCOR2
SCHEMBL3235296 0.77 HDAC1 (0.70) HDAC3HDAC1HDAC2HDAC10NCOR2
SCHEMBL3238723 0.75 HDAC1 (0.61) HDAC3HDAC1HDAC2HDAC10NCOR2
SCHEMBL7929398 0.74 HDAC1 (0.74) HDAC3HDAC1HDAC2HDAC10NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO claimed
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed