SCHEMBL3236170

SCHEMBL3236170

O=C(O)c1nccc(Nc2ccccc2)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 10/20 0.61
AURKB Q96GD4 3/20 0.61
RAB9A P51151 3/20 0.59
NPC1 O15118 2/20 0.59
MAPT P10636 2/20 0.59
CHEK1 O14757 1/20 0.59
IKBKB O14920 1/20 0.59
PDPK1 O15530 1/20 0.59
CHEK2 O96017 1/20 0.59
PRKCG P05129 1/20 0.59
CDK1 P06493 1/20 0.59
LYN P07948 1/20 0.59
KIT P10721 1/20 0.59
PIM1 P11309 1/20 0.59
FGFR1 P11362 1/20 0.59
FGFR3 P22607 1/20 0.59
RPS6KB1 P23443 1/20 0.59
CDK2 P24941 1/20 0.59
MARK3 P27448 1/20 0.59
MAPK1 P28482 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25884869 0.87 AURKA (0.56) AURKAAURKBRAB9ANPC1MAPT
SCHEMBL29448928 0.87 AURKA (0.60) AURKAAURKBRAB9ANPC1MAPT
SCHEMBL30748867 0.87 AURKA (0.52) AURKAAURKBRAB9ANPC1MAPT
SCHEMBL31480553 0.77 HCAR3 (0.46) AURKAHCAR3
SCHEMBL4884433 0.77 AURKA (0.65) AURKAAURKBRAB9ANPC1MAPT
Hydrochloric Acid SCHEMBL15487562 0.75 AURKA (0.97) AURKAAURKBRAB9ANPC1MAPT
SCHEMBL30748839 0.75 SCN9A (0.50) AURKAAURKBRAB9ANPC1MAPT
SCHEMBL31691345 0.74 ROCK1 (0.51) AURKAAURKBRAB9ANPC1MAPT
SCHEMBL440486 0.74 AURKA (1.00) AURKAAURKBRAB9ANPC1MAPT
SCHEMBL3988183 0.73 AURKA (0.65) AURKAAURKBRAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4215526-A1 CARBONYL HETEROCYCLIC COMPOUND AND APPLICATION THEREOF Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2023-07-26 EP disclosed
WO-2010020432-A8 COMPOUNDS FOR TREATMENT OF DUCHENNE MUSCULAR DYSTROPHY BIOMARIN IGA LIMITED (BS) 2010-03-11 WO disclosed
WO-2010020432-A2 COMPOUNDS FOR TREATMENT OF DUCHENNE MUSCULAR DYSTROPHY SUMMIT CORPORATION PLC (GB) 2010-02-25 WO disclosed