SCHEMBL3236708

SCHEMBL3236708

Cc1cc(C)c(C(=O)NC(c2ccccc2)C2(N(C)C)CCCC2)c(C)c1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 16/20 0.48
SLC6A5 Q9Y345 1/20 0.46
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TAS1R3 Q7RTX0 2/20 0.37
TAS1R1 Q7RTX1 2/20 0.37
TAS1R2 Q8TE23 2/20 0.37
PYGL P06737 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3243915 0.91 SLC6A9 (0.47) SLC6A9SLC6A5
SCHEMBL3237783 0.91 SLC6A9 (0.47) SLC6A9SLC6A5
SCHEMBL3230781 0.90 SLC6A9 (0.59) SLC6A9SLC6A5
SCHEMBL13780494 0.90 SLC6A9 (0.59) SLC6A9SLC6A5
SCHEMBL3230762 0.89 SLC6A9 (0.45) SLC6A9SLC6A5MEN1KMT2A
SCHEMBL3239525 0.86 UTS2R (0.43) SLC6A9SLC6A5KMT2ASMN1; SMN2TAS1R3
SCHEMBL3037837 0.84 SLC6A9 (0.47) SLC6A9SLC6A5
SCHEMBL3034321 0.84 SLC6A9 (0.49) SLC6A9SLC6A5
SCHEMBL3239596 0.83 CNR1 (0.41) SLC6A9SLC6A5MEN1KMT2APYGL
SCHEMBL13303986 0.83 SLC6A9 (0.41) SLC6A9SLC6A5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745642-B2 Glycine transport inhibitors GLAXO GROUP LIMITED (GB) 2010-06-29 US disclosed
US-7745642-B2 Glycine transport inhibitors GLAXO GROUP LIMITED (GB) 2010-06-29 US disclosed
US-7745642-B2 Glycine transport inhibitors GLAXO GROUP LIMITED (GB) 2010-06-29 US disclosed
US-20080287547-A1 Glycine Transport Inhibitors GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed
US-20080287547-A1 Glycine Transport Inhibitors GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed
US-20080287547-A1 Glycine Transport Inhibitors GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080287547-A1 Glycine Transport Inhibitors SLC18A2, SLC6A5, SLC1A2 SLC6A9 13/4885SLC6A5 2/4885MEN1 2501/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.