SCHEMBL3236751

SCHEMBL3236751

COc1ccc2c(c1)CN(C(=O)Cn1c(=O)n(C)c3cc(-c4cc(Cl)cc(Cl)c4)cnc31)CC2

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 19/20 0.46
GRIN2B Q13224 19/20 0.46
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3245549 0.97 GRIN1 (0.46) GRIN1GRIN2BADORA2AADORA2BADORA1
SCHEMBL3242733 0.93 GRIN1 (0.50) GRIN1GRIN2B
SCHEMBL3247379 0.88 GRIN1 (0.51) GRIN1GRIN2BADORA2AADORA2BADORA1
SCHEMBL3245322 0.88 GRIN1 (0.51) GRIN1GRIN2B
SCHEMBL3249233 0.86 GRIN2B (0.61) GRIN1GRIN2B
SCHEMBL3252047 0.86 GRIN1 (0.46) GRIN1GRIN2B
SCHEMBL3252351 0.83 GRIN2B (0.52) GRIN1GRIN2B
SCHEMBL13521617 0.82 GRIN1 (0.58) GRIN1GRIN2B
SCHEMBL13521708 0.80 GRIN1 (0.63) GRIN1GRIN2B
SCHEMBL3256125 0.79 GRIN2B (0.55) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO claimed
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed