SCHEMBL3237306

SCHEMBL3237306

CCCNc1ccc(C(=O)NC2CCCCC2)c(SCCC)n1

nearest known ligand 0.84

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 20/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2007008 0.92 HSD11B1 (1.00) HSD11B1
SCHEMBL13182824 0.90 HSD11B1 (0.85) HSD11B1
SCHEMBL1971515 0.85 HSD11B1 (1.00) HSD11B1
SCHEMBL12571009 0.85 HSD11B1 (1.00) HSD11B1
SCHEMBL2008255 0.84 HSD11B1 (0.67) HSD11B1
SCHEMBL2008865 0.84 HSD11B1 (0.83) HSD11B1
SCHEMBL12571587 0.84 HSD11B1 (0.83) HSD11B1
SCHEMBL1972941 0.83 HSD11B1 (1.00) HSD11B1
SCHEMBL12571013 0.83 HSD11B1 (1.00) HSD11B1
SCHEMBL3401955 0.83 HSD11B1 (0.76) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233480-B1 Chemical compounds ASTRAZENECA AB (SE) 2013-05-29 EP disclosed
EP-2233480-A1 Chemical compounds AstraZeneca AB (SE) 2010-09-29 EP disclosed
EP-2086939-B1 PYRIDINE CARBOXAMIDES AS 11-BETA-HSD1 INHIBITORS ASTRAZENECA AB (SE) 2010-07-28 EP disclosed