SCHEMBL3239092

SCHEMBL3239092

COc1ccc2c(c1)CN(C(=O)CN1C(=O)CCc3cc(-c4ccc(F)c(Cl)c4)cnc31)C2

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 16/20 0.43
ROCK1 Q13464 1/20 0.39
HSD17B3 P37058 1/20 0.38
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
MAPK1 P28482 1/20 0.37
GRIN1 Q05586 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3124617 0.94 GRIN2B (0.42) GRIN2BHSD17B3ESR1ESR2MAPK1
SCHEMBL13521688 0.90 GRIN2B (0.41) GRIN2B
SCHEMBL3247392 0.89 HSD17B3 (0.43) GRIN2BROCK1HSD17B3ESR1ESR2
SCHEMBL3239090 0.85 GRIN2B (0.41) GRIN2BGRIN1
SCHEMBL3264528 0.85 MAPK1 (0.44) GRIN2BHSD17B3ESR1ESR2MAPK1
SCHEMBL3128418 0.85 ROCK1 (0.37) ROCK1HSD17B3ESR1ESR2MAPK1
SCHEMBL3118590 0.84 ESR2 (0.45) ESR1ESR2MAPK1
SCHEMBL3127545 0.84 MAPK1 (0.41) ESR1ESR2MAPK1
SCHEMBL13521598 0.83 HSD17B3 (0.43) GRIN2BHSD17B3ESR1ESR2MAPK1
SCHEMBL3127648 0.83 GAA (0.43) GRIN2BESR2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO claimed
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO disclosed