SCHEMBL3239722

SCHEMBL3239722

COC(=O)Oc1ccc(C(=O)c2ccccc2F)o1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.42
ALDH1A1 P00352 5/20 0.42
HPGD P15428 4/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
MEN1 O00255 2/20 0.38
MAPT P10636 2/20 0.38
HTT P42858 1/20 0.38
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
KAT6A Q92794 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3239963 0.84 ALDH1A1 (0.43) KMT2AALDH1A1HPGDGAASMN1; SMN2
SCHEMBL5371049 0.80 KMT2A (0.49) KMT2AALDH1A1HPGDHSD17B10KDM4E
SCHEMBL3240065 0.78 ALDH1A1 (0.38) KMT2AALDH1A1HPGDGAASMN1; SMN2
SCHEMBL3241870 0.78 ALDH1A1 (0.40) KMT2AALDH1A1HPGDKDM4EGAA
SCHEMBL3241897 0.76 ALDH1A1 (0.41) KMT2AALDH1A1HPGDHSD17B10KDM4E
SCHEMBL1439154 0.73 HSD17B10 (0.42) KMT2AALDH1A1HPGDHSD17B10KDM4E
SCHEMBL3239957 0.72 ALDH1A1 (0.49) KMT2AALDH1A1HPGDGAANPC1
SCHEMBL30293901 0.67 CES2 (0.71) KMT2AALDH1A1HPGDGAANPC1
SCHEMBL250099 0.67 CES2 (0.71) KMT2AALDH1A1HPGDGAANPC1
SCHEMBL15454164 0.67 HPGD (0.59) KMT2AALDH1A1HPGDHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1418176-B1 Pyrazole derivates, their preparation and their use in drugs SANOFI AVENTIS DEUTSCHLAND (DE) 2010-04-28 EP disclosed
EP-1418176-A1 Pyrazole derivates, their preparation and their use in drugs Aventis Pharma Deutschland GmbH (DE) 2004-05-12 EP disclosed
EP-0908456-B1 Pyrazole derivatives, their preparation and their use in drugs AVENTIS PHARMA GMBH (DE) 2003-12-17 EP disclosed
EP-0908456-A1 Pyrazole derivatives, their preparation and their use in drugs Hoechst Marion Roussel Deutschland GmbH (DE) 1999-04-14 EP disclosed