SCHEMBL3240712

SCHEMBL3240712

O=C=Nc1cccc(I)c1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
NOTUM Q6P988 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
TRPA1 O75762 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1493080 0.87 CYP3A4 (0.54) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL1161021 0.80 CYP3A4 (0.47) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL4242346 0.80 CYP3A4 (0.47) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL1133625 0.79 CYP3A4 (0.46) CYP3A4NOTUMGABRA1GABRB2TRPA1
SCHEMBL964183 0.79 CYP3A4 (0.55) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL3453793 0.75 CYP3A4 (0.46) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL93319 0.74 CYP3A4 (0.52) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL25147648 0.73 NOTUM (0.44) NOTUM
SCHEMBL11872591 0.72 CYP3A4 (0.56) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL3399383 0.72 CYP3A4 (0.73) CYP3A4GABRA1GABRB2TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010011917-A1 SEH AND 11β-HSD1 DUAL INHIBITORS GLAXOSMITHKLINE LLC (US) 2010-01-28 WO disclosed