SCHEMBL4242346

SCHEMBL4242346

O=C=Nc1cccc(C(F)(F)F)c1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.47
HSD11B1 P28845 1/20 0.34
PARP1 P09874 1/20 0.33
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
CES1 P23141 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KDM4E B2RXH2 2/20 0.31
NOS3 P29474 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1493080 0.88 CYP3A4 (0.54) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL75112 0.82 CYP3A4 (0.47) CYP3A4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL29648814 0.82 CYP3A4 (0.47) CYP3A4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL1513863 0.81 CYP3A4 (0.47) CYP3A4PARP1GABRA1GABRB2KDM4E
SCHEMBL29648824 0.81 CYP3A4 (0.47) CYP3A4PARP1GABRA1GABRB2GRIN2D
SCHEMBL59215 0.81 CYP3A4 (0.47) CYP3A4PARP1GABRA1GABRB2GRIN2D
SCHEMBL7062055 0.81 ALDH1A1 (0.47) CYP3A4HSD11B1GABRA1GABRB2GRIN2D
SCHEMBL1161021 0.81 CYP3A4 (0.47) CYP3A4GABRA1GABRB2TRPA1
SCHEMBL3460968 0.80 CYP3A4 (0.66) CYP3A4HSD11B1PARP1GABRA1GABRB2
SCHEMBL1133625 0.80 CYP3A4 (0.46) CYP3A4GABRA1GABRB2TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111100732-B Soap urethane lubricating grease and preparation method thereof 中国石油化工股份有限公司 2022-10-21 CN claimed
CN-111100732-A Soap urethane lubricating grease and preparation method thereof 中国石油化工股份有限公司 2020-05-05 CN claimed
CN-109804487-A The electrolyte comprising additive for high-energy rechargeable metal anode battery 派立昂技术公司 2019-05-24 CN claimed
CN-109354662-A Anti-infection material for built-in hemodialysis tube and preparation method thereof 湖南博隽生物医药有限公司 2019-02-19 CN claimed
US-20090216006-A1 COVALENTLY BOUND POLYSACCHARIDE-BASED CHIRAL STATIONARY PHASES AND METHOD FOR THEIR PREPARATION XU HUI 2009-08-27 US claimed
CN-111100732-B Soap urethane lubricating grease and preparation method thereof 中国石油化工股份有限公司 2022-10-21 CN disclosed
CN-111100732-A Soap urethane lubricating grease and preparation method thereof 中国石油化工股份有限公司 2020-05-05 CN disclosed
CN-109804487-A The electrolyte comprising additive for high-energy rechargeable metal anode battery 派立昂技术公司 2019-05-24 CN disclosed
CN-109608513-A 18 β-enoxolone carbamate derivatives and its preparation method and application 锦州医科大学 2019-04-12 CN disclosed
CN-109354662-A Anti-infection material for built-in hemodialysis tube and preparation method thereof 湖南博隽生物医药有限公司 2019-02-19 CN disclosed
WO-2008067222-A1 HETEROCYCLIC MODULATORS OF TGR5 KALYPSYS, INC. (US) 2008-06-05 WO disclosed
EP-1608373-A2 TIE-2 MODULATORS AND METHODS OF USE Exelixis Inc. (US) 2005-12-28 EP disclosed
EP-1558582-A1 DIARYL AND ARYLHETEROARYL UREA DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE PROPHYLAXIS AND TREATMENT OF DISORDERS RELATED THERETO Arena Pharmaceuticals, Inc. (US) 2005-08-03 EP disclosed
WO-2005012254-A1 DIARYL AND ARYLHETEROARYL UREA DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE PROPHYLAXIS AND TREATMENT OF DISORDERS RELATED THERTO ARENA PHARMACEUTICALS, INC. (US) 2005-02-10 WO disclosed
WO-2004083235-A2 TIE-2 MODULATORS AND METHODS OF USE EXELIXIS INC. (US) 2004-09-30 WO disclosed
US-6316623-B1 USEFUL FOR SCREENING IN BIOLOGICAL ASSAYS IN ORDER TO IDENTIFY PHARMACEUTICALLY USEFUL COMPOUNDS ISIS PHARMACEUTICALS, INC. 2001-11-13 US disclosed