SCHEMBL3241071

SCHEMBL3241071

COc1cccc([C@@]2(C)CC3(N=C(SC)NC3=O)c3cc(Br)ccc3O2)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 8/20 0.39
CTSD P07339 7/20 0.39
HCAR2 Q8TDS4 1/20 0.34
HSP90AA1 P07900 2/20 0.34
APP P05067 1/20 0.33
MEN1 O00255 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HIF1A Q16665 1/20 0.32
CXCR3 P49682 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
HSD11B1 P28845 1/20 0.32
LMNA P02545 1/20 0.31
TP53 P04637 2/20 0.31
MDM2 Q00987 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1831618 0.87 BACE1 (0.39) BACE1CTSDHCAR2HSD11B1
SCHEMBL1827904 0.81 BACE1 (0.40) BACE1CTSDHCAR2
SCHEMBL1829080 0.80 BACE1 (0.39) BACE1CTSD
SCHEMBL1829335 0.74 BACE1 (0.44) BACE1CTSDHCAR2HSD11B1
SCHEMBL1826421 0.74 BACE1 (0.47) BACE1CTSDHSD11B1
SCHEMBL1828227 0.73 BACE1 (0.40) BACE1CTSDAPPCYP3A4CYP2C19
SCHEMBL2375695 0.69 BACE1 (0.54) BACE1CTSD
SCHEMBL2376232 0.69 BACE1 (0.54) BACE1CTSD
SCHEMBL2375445 0.69 BACE1 (0.54) BACE1CTSD
SCHEMBL12246431 0.69 BACE1 (0.50) BACE1CTSDKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed