SCHEMBL3241853

SCHEMBL3241853

Nc1ccc(F)cc1NC(=O)CCCCCC(=O)NCc1cccs1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.61
HDAC3 O15379 10/20 0.57
HDAC1 Q13547 9/20 0.57
MAPK1 P28482 2/20 0.51
TP53 P04637 1/20 0.51
ALOX15 P16050 1/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
HSD17B10 Q99714 1/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
TSHR P16473 1/20 0.48
HDAC2 Q92769 2/20 0.46
HPGD P15428 2/20 0.46
ALDH1A1 P00352 2/20 0.46
NCOR2 Q9Y618 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7925289 0.85 USP2 (0.68) USP2HDAC3HDAC1POLBMAPT
SCHEMBL7940673 0.80 USP2 (0.52) USP2MAPK1TP53ALOX15CASP1
SCHEMBL17009233 0.77 USP2 (0.85) USP2MAPK1TP53ALOX15CASP1
SCHEMBL7694996 0.77 USP2 (0.85) USP2MAPK1TP53ALOX15CASP1
SCHEMBL3238234 0.76 HDAC1 (0.70) HDAC3HDAC1HDAC2NCOR2HDAC4
SCHEMBL17009271 0.76 USP2 (0.88) USP2MAPK1TP53ALOX15CASP1
SCHEMBL3240756 0.76 HDAC3 (0.59) USP2HDAC3HDAC1MAPK1TP53
SCHEMBL13438260 0.75 USP2 (0.93) USP2MAPK1TP53ALOX15CASP1
SCHEMBL12472765 0.74 KDM4E (0.48) USP2MAPK1MEN1KMT2APOLB
SCHEMBL9784530 0.73 USP2 (0.82) USP2MAPK1TP53ALOX15CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO disclosed