SCHEMBL3244269

SCHEMBL3244269

CCCC1=C(C(=O)OCC)C(c2ccsc2)C2=C(CC(C(C)C)CC2=O)N1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 12/20 0.55
ALDH1A1 P00352 8/20 0.55
HSD17B10 Q99714 6/20 0.55
HPGD P15428 4/20 0.55
CASP1 P29466 5/20 0.51
POLB P06746 5/20 0.51
CASP7 P55210 4/20 0.51
LMNA P02545 2/20 0.49
ADORA2B P29275 7/20 0.46
USP2 O75604 1/20 0.45
TSHR P16473 1/20 0.45
RAB9A P51151 1/20 0.42
AGTR1 P30556 1/20 0.42
GAA P10253 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MCL1 Q07820 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3003468 0.83 KDM4E (0.79) KDM4EALDH1A1HSD17B10HPGDCASP1
SCHEMBL3250423 0.83 KDM4E (0.79) KDM4EALDH1A1HSD17B10HPGDCASP1
SCHEMBL3008977 0.81 KDM4E (0.55) KDM4EALDH1A1HSD17B10HPGDCASP1
SCHEMBL13521836 0.73 KDM4E (0.66) KDM4EALDH1A1HSD17B10HPGDCASP1
SCHEMBL13096488 0.73 KDM4E (0.69) KDM4EALDH1A1HSD17B10HPGDCASP1
SCHEMBL3005577 0.71 KDM4E (1.00) KDM4EALDH1A1HSD17B10HPGDCASP1
SCHEMBL6461607 0.70 KDM4E (0.73) KDM4EALDH1A1HSD17B10HPGDCASP1
SCHEMBL5333713 0.69 KDM4E (0.65) KDM4EALDH1A1HSD17B10HPGDCASP1
SCHEMBL5823841 0.69 HTR1A (0.48) KDM4EALDH1A1HSD17B10HPGDCASP1
SCHEMBL5816717 0.68 HTR1A (0.60) KDM4EALDH1A1HSD17B10HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010002483-A1 OPTIONALLY CONDENSED DIHYDRO PYRIDINE, DIHYDROPYRIMIDINE AND DIHYDRO PYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2010-01-07 WO disclosed
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed