SCHEMBL3244351

SCHEMBL3244351

CC(C)(C)OC(=O)NC1CC[C@H](S(=O)(=O)c2cc3c(cc2Cl)[nH]c(=O)c2[nH]cc(C(=O)O)c23)C1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BTK Q06187 8/20 0.40
KAT6A Q92794 1/20 0.39
KAT5 Q92993 1/20 0.39
JAK1 P23458 4/20 0.33
JAK2 O60674 2/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
KAT8 Q9H7Z6 4/20 0.33
KDM1A O60341 1/20 0.32
MAOB P27338 1/20 0.32
MAPK8 P45983 1/20 0.32
DDR1 Q08345 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244356 1.00 BTK (0.40) BTKKAT6AKAT5JAK1JAK2
SCHEMBL4173768 0.86 KAT6A (0.35) BTKKAT6AKAT5KAT8MAPK8
Butyric Acid SCHEMBL4173769 0.81 KAT6A (0.38) BTKKAT6AKAT5JAK1JAK2
Hydrochloric Acid SCHEMBL3250727 0.81 CSNK2A2 (0.32) BTK
Hydrochloric Acid SCHEMBL3250722 0.81 CSNK2A2 (0.32) BTK
SCHEMBL3242979 0.74 KDM4E (0.45) JAK1JAK2JAK3
SCHEMBL3242728 0.74 KDM4E (0.45) JAK1JAK2JAK3
SCHEMBL3242729 0.74 KDM4E (0.45) JAK1JAK2JAK3
SCHEMBL3254879 0.72 PRKAG1 (0.40)
SCHEMBL4159322 0.66 CCR8 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP disclosed