SCHEMBL3393346

SCHEMBL3393346

COc1ccccc1-c1cnnc(N)n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.59
HSP90AB1 P08238 1/20 0.57
ALDH1A1 P00352 4/20 0.50
GAA P10253 2/20 0.50
MAPT P10636 1/20 0.50
HPGD P15428 1/20 0.50
ALOX15 P16050 1/20 0.50
ALOX12 P18054 1/20 0.50
HSD17B10 Q99714 1/20 0.50
ATR Q13535 2/20 0.48
METAP2 P50579 1/20 0.47
ADORA2A P29274 4/20 0.47
KDM4E B2RXH2 1/20 0.46
PTPN1 P18031 1/20 0.46
ADORA1 P30542 2/20 0.46
JAK2 O60674 1/20 0.44
CHRNA7 P36544 1/20 0.44
ATP4A P20648 1/20 0.43
ATP4B P51164 1/20 0.43
DHFR P00374 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13425400 0.86 GAA (0.50) HSP90AA1HSP90AB1ALDH1A1GAAMAPT
SCHEMBL3399496 0.83 CHRNA7 (0.47) HSP90AA1HSP90AB1ALDH1A1GAAMAPT
SCHEMBL3397291 0.83 MAOB (0.47) HSP90AA1HSP90AB1ALDH1A1ADORA2AADORA1
SCHEMBL3246149 0.82 HSP90AA1 (0.56) HSP90AA1HSP90AB1ALDH1A1ADORA2AKDM4E
SCHEMBL3394031 0.81 NCOA1 (0.44) HSP90AA1HSP90AB1ATRADORA2AADORA1
SCHEMBL3398117 0.80 MPL (0.44) HSP90AA1MAPTADORA2AKDM4EADORA1
SCHEMBL3395005 0.80 DHFR (0.47) HSP90AA1HSP90AB1ALDH1A1MAPTHPGD
SCHEMBL3393510 0.80 ADORA2A (0.40) HSP90AA1HSP90AB1ATRADORA2AADORA1
SCHEMBL13425651 0.80 CYP1A2 (0.49)
SCHEMBL27990113 0.78 ALDH1A1 (0.51) HSP90AA1HSP90AB1ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102822150-B 1,2, 4-triazin-4-amine derivatives HEPTARES THERAPEUTICS LTD 2014-12-03 CN disclosed
CN-102822150-A 1,2, 4-triazin-4-amine derivatives HEPTARES THERAPEUTICS LTD 2012-12-12 CN disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed