SCHEMBL3247175

SCHEMBL3247175

COc1cccc(COC(=O)Nc2cc(F)c(-c3cn[nH]c3)cc2OCCCO)c1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 18/20 0.57
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
ROCK1 Q13464 5/20 0.51
CDC42BPA Q5VT25 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3245071 0.91 ROCK2 (0.69) ROCK2NPC1RAB9AROCK1CDC42BPA
SCHEMBL3239562 0.87 ROCK2 (0.59) ROCK2ROCK1
SCHEMBL3239731 0.87 ROCK2 (0.60) ROCK2NPC1RAB9AROCK1CDC42BPA
SCHEMBL3248264 0.83 ROCK2 (0.62) ROCK2NPC1RAB9AROCK1CDC42BPA
SCHEMBL3252352 0.80 ROCK2 (0.64) ROCK2ROCK1CDC42BPA
SCHEMBL3253611 0.79 ROCK2 (0.61) ROCK2NPC1RAB9AROCK1CDC42BPA
SCHEMBL13391213 0.78 ROCK2 (0.71) ROCK2ROCK1CDC42BPA
SCHEMBL3238586 0.77 ROCK2 (0.52) ROCK2ROCK1CDC42BPA
SCHEMBL3255470 0.77 ROCK2 (0.74) ROCK2ROCK1CDC42BPA
SCHEMBL3247183 0.76 ROCK2 (0.53) ROCK2ROCK1CDC42BPA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed