SCHEMBL3247331

SCHEMBL3247331

O=C(OCc1ccc2c(c1)OCCO2)N(CCO)c1ccc(-c2cn[nH]c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 14/20 0.51
CYP3A4 P08684 2/20 0.38
ROCK1 Q13464 5/20 0.38
PTGES O14684 1/20 0.38
ALOX5 P09917 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CDC42BPA Q5VT25 1/20 0.38
FAAH O00519 1/20 0.36
MGLL Q99685 1/20 0.36
NPC1 O15118 1/20 0.36
ALPL P05186 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3244974 0.79 ROCK2 (0.65) ROCK2ROCK1FAAHMAPT
SCHEMBL3241276 0.78 ROCK2 (0.72) ROCK2CYP3A4ROCK1CYP2D6CYP2C9
SCHEMBL3265254 0.78 ROCK2 (0.53) ROCK2CYP3A4ROCK1CYP2D6CYP2C9
SCHEMBL3265256 0.76 ROCK2 (0.53) ROCK2CYP3A4ROCK1CYP2D6CYP2C9
SCHEMBL3252994 0.74 ROCK2 (0.49) ROCK2CYP3A4ROCK1CYP2D6CYP2C9
SCHEMBL3242441 0.74 ROCK2 (0.49) ROCK2CYP3A4ROCK1CYP2D6CYP2C9
SCHEMBL3244390 0.74 ROCK2 (0.50) ROCK2CYP3A4ROCK1CYP2D6CYP2C9
SCHEMBL3244090 0.73 ROCK2 (0.65) ROCK2CYP3A4ROCK1CYP2D6CYP2C9
SCHEMBL3264992 0.72 ROCK2 (0.72) ROCK2CYP3A4ROCK1CYP2D6CYP2C9
SCHEMBL3253893 0.71 ROCK1 (0.55) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed