SCHEMBL3247611

SCHEMBL3247611

COc1cc(OC)cc(S(=O)(=O)NCC(=O)Nc2ccc(Cl)cc2Cc2ccccc2Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
MEP1B Q16820 1/20 0.44
ALDH1A1 P00352 6/20 0.43
LMNA P02545 2/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 3/20 0.42
KDM4E B2RXH2 2/20 0.42
GAA P10253 2/20 0.42
HPGD P15428 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
OXTR P30559 1/20 0.41
AVPR1A P37288 1/20 0.41
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41
KDR P35968 1/20 0.41
MAPK1 P28482 2/20 0.41
HTT P42858 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3255565 0.93 MEP1B (0.55) TSHRMEP1BALDH1A1LMNAPOLB
SCHEMBL3253721 0.92 TSHR (0.48) TSHRMEP1BALDH1A1POLBMAPT
SCHEMBL3251190 0.87 ALDH1A1 (0.46) TSHRALDH1A1LMNAMAPTKDM4E
SCHEMBL3249160 0.87 ALDH1A1 (0.53) TSHRMEP1BALDH1A1LMNAPOLB
SCHEMBL3253246 0.87 MEP1B (0.48) TSHRMEP1BALDH1A1LMNAMAPT
SCHEMBL3247755 0.87 MAPK1 (0.59) TSHRMEP1BALDH1A1LMNAMAPT
SCHEMBL3253380 0.85 MAPT (0.52) TSHRALDH1A1LMNAMAPTKDM4E
SCHEMBL3251138 0.85 GAA (0.47) TSHRALDH1A1LMNAMAPTKDM4E
SCHEMBL3255473 0.84 ALDH1A1 (0.47) TSHRMEP1BALDH1A1LMNAPOLB
SCHEMBL3255588 0.84 TSHR (0.46) TSHRMEP1BALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776347-B1 SULPHONAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION SANOFI AVENTIS (FR) 2010-05-26 EP disclosed