SCHEMBL3247658

SCHEMBL3247658

O=CCN1CCC(C(=NO)c2ccc(Cl)cc2Cl)CC1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A12 P48065 1/20 0.41
NOTUM Q6P988 2/20 0.40
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39
ALOX15 P16050 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ACKR3 P25106 1/20 0.37
OGG1 O15527 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
HIF1A Q16665 1/20 0.35
SRD5A2 P31213 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10634934 0.84 NOTUM (0.42) SLC6A12NOTUMUSP2LMNAALOX15
SCHEMBL3240425 0.84 SLC6A12 (0.46) SLC6A12NOTUMACKR3ALDH1A1MAPK1
Formic Acid SCHEMBL10640837 0.81 NOTUM (0.40) SLC6A12NOTUMUSP2LMNAALOX15
SCHEMBL7503531 0.78 HTR2A (0.39) MEN1KMT2AACKR3ALDH1A1
SCHEMBL606330 0.78 MEN1 (0.47) NOTUMHRH4MEN1KMT2AALDH1A1
SCHEMBL606329 0.78 MEN1 (0.47) NOTUMHRH4MEN1KMT2AALDH1A1
SCHEMBL10634910 0.74 KMT2A (0.47) NOTUMUSP2LMNAALOX15HRH4
SCHEMBL21381592 0.74 CPS1 (0.44) MEN1KMT2AACKR3ALDH1A1
Hydrochloric Acid SCHEMBL10634903 0.73 KMT2A (0.46) NOTUMUSP2LMNAALOX15HRH4
SCHEMBL4983350 0.72 HSD11B1 (0.55) MEN1KMT2AACKR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183245-A2 DUAL MODULATORS OF 5-HT2A AND D3 RECEPTORS F. Hoffmann-Roche AG (CH) 2010-05-12 EP disclosed
WO-2009013212-A2 DUAL MODULATORS OF 5-HT2A AND D3 RECEPTORS F. HOFFMANN-LA ROCHE AG (CH) 2009-01-29 WO disclosed