SCHEMBL3248160

SCHEMBL3248160

CCCCCc1cnnc(Cl)n1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.44
CYP19A1 P11511 7/20 0.36
GABRA2 P47869 2/20 0.35
GABRB2 P47870 2/20 0.35
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MIF P14174 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GPR84 Q9NQS5 1/20 0.33
KMT2A Q03164 1/20 0.33
NOS2 P35228 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11117895 0.79 KCNH2 (0.46) KCNH2CYP19A1TDP1L3MBTL1MIF
SCHEMBL2359176 0.78 KCNH2 (0.44) KCNH2TDP1L3MBTL1KMT2ANOS2
SCHEMBL426455 0.76 KCNH2 (0.50) KCNH2CYP19A1GABRA2GABRB2GPR84
SCHEMBL22616936 0.76 KCNH2 (0.46) KCNH2CYP19A1GABRA2GABRB2TDP1
SCHEMBL2364044 0.75 MAPT (0.43) KCNH2TDP1L3MBTL1MIFCYP2C9
SCHEMBL12539240 0.75 KCNH2 (0.53) KCNH2CYP19A1GABRA2GABRB2GPR84
SCHEMBL2364312 0.73 KCNH2 (0.40) KCNH2CYP19A1TDP1L3MBTL1MIF
SCHEMBL791579 0.72 KCNH2 (0.46) KCNH2CYP19A1GABRA2GABRB2GPR84
SCHEMBL10830973 0.71 KCNH2 (0.44) KCNH2CYP19A1TDP1L3MBTL1MIF
SCHEMBL4301655 0.70 KCNH2 (0.53) KCNH2CYP19A1TDP1L3MBTL1MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001220-A1 NEW 1,2,4-TRIAZINE DERIVATIVES AND BIOLOGICAL APPLICATIONS THEREOF MUTABILIS SA (FR) 2010-01-07 WO disclosed
EP-2141164-A1 New 1,2,4-triazine derivatives and biological applications thereof Mutabilis (FR) 2010-01-06 EP disclosed