SCHEMBL3249509

SCHEMBL3249509

CC1=C(C(=O)NCCCCc2ccccc2)C(c2ccsc2)C2=C(CCCC2=O)N1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.61
HSD17B10 Q99714 5/20 0.61
CASP1 P29466 2/20 0.61
ALDH1A1 P00352 9/20 0.60
HPGD P15428 8/20 0.60
SMN1; SMN2 Q16637 2/20 0.54
KMT2A Q03164 1/20 0.54
RAB9A P51151 1/20 0.52
FFAR3 O14843 8/20 0.51
GLA P06280 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TSHR P16473 1/20 0.46
ALOX12 P18054 1/20 0.46
LMNA P02545 3/20 0.46
CASP7 P55210 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3000122 0.78 KDM4E (0.69) KDM4EHSD17B10CASP1ALDH1A1HPGD
SCHEMBL3005577 0.75 KDM4E (1.00) KDM4EHSD17B10CASP1ALDH1A1HPGD
SCHEMBL3242208 0.73 FFAR3 (0.70) KDM4EHSD17B10CASP1ALDH1A1HPGD
SCHEMBL3002415 0.73 KDM4E (0.77) KDM4EHSD17B10CASP1ALDH1A1HPGD
SCHEMBL3007058 0.73 KDM4E (0.74) KDM4EHSD17B10CASP1ALDH1A1HPGD
SCHEMBL3003468 0.69 KDM4E (0.79) KDM4EHSD17B10CASP1ALDH1A1HPGD
SCHEMBL3329777 0.68 ALDH1A1 (0.78) KDM4EHSD17B10CASP1ALDH1A1HPGD
SCHEMBL16211041 0.68 SMN1; SMN2 (0.73) KDM4EHSD17B10CASP1ALDH1A1HPGD
SCHEMBL3324655 0.68 SMN1; SMN2 (0.72) KDM4EHSD17B10CASP1ALDH1A1HPGD
SCHEMBL12784576 0.67 ALDH1A1 (0.64) KDM4EHSD17B10CASP1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010002483-A1 OPTIONALLY CONDENSED DIHYDRO PYRIDINE, DIHYDROPYRIMIDINE AND DIHYDRO PYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2010-01-07 WO disclosed
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed