SCHEMBL325009

SCHEMBL325009

FC(F)(F)c1cccc(C(c2nnn[nH]2)N2CCOCC2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.61
KMT2A Q03164 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.44
OPRL1 P41146 4/20 0.43
OPRM1 P35372 3/20 0.43
OPRD1 P41143 3/20 0.43
OPRK1 P41145 3/20 0.43
RECQL P46063 1/20 0.42
LMNA P02545 2/20 0.41
CNR2 P34972 1/20 0.41
CACNA2D1 P54289 1/20 0.41
CACNA1B Q00975 1/20 0.41
CACNB1 Q02641 1/20 0.41
CACNA1C Q13936 1/20 0.41
CHRM2 P08172 1/20 0.39
HTR1A P08908 1/20 0.39
DRD3 P35462 1/20 0.39
HTR2B P41595 1/20 0.39
MIF P14174 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL324720 0.99 ALDH1A1 (0.60) ALDH1A1KMT2AL3MBTL1OPRL1OPRM1
SCHEMBL12503128 0.77 ALDH1A1 (0.39) ALDH1A1KMT2ALMNAMIFGAA
SCHEMBL325375 0.76 SLC6A2 (0.45) ALDH1A1KMT2AL3MBTL1LMNACNR2
SCHEMBL325002 0.74 ALDH1A1 (0.47) ALDH1A1KMT2ACHRM2HTR1ADRD3
SCHEMBL11158619 0.70 RPS6KB1 (0.54) ALDH1A1KMT2AL3MBTL1LMNACNR2
SCHEMBL4152093 0.70 SLC6A4 (0.60) ALDH1A1KMT2AOPRL1OPRM1OPRD1
Hydrochloric Acid SCHEMBL14815137 0.69 ALDH1A1 (0.52) ALDH1A1KMT2AL3MBTL1OPRL1OPRM1
SCHEMBL4575599 0.68 IDO1 (0.43) KMT2AOPRM1OPRK1LMNACACNA1C
SCHEMBL4135481 0.67 MEN1 (0.66) ALDH1A1KMT2AOPRL1OPRM1OPRD1
SCHEMBL1281621 0.66 MEN1 (0.65) KMT2AOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590953-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2013-05-15 EP claimed
WO-2012004604-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2012-01-12 WO claimed
EP-2590953-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2013-05-15 EP disclosed
WO-2012004604-A1 TETRAZOLE COMPOUNDS AS CALCIUM CHANNEL BLOCKERS Convergence Pharmaceuticals Limited (GB) 2012-01-12 WO disclosed