SCHEMBL3250686

SCHEMBL3250686

CCOC(=O)Oc1c[nH]c2c(=O)[nH]c3ccc(S(=O)(=O)NC4CCCCC4)cc3c12

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.52
LMNA P02545 4/20 0.45
ALDH1A1 P00352 4/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
GAA P10253 3/20 0.45
THRB P10828 1/20 0.45
PARG Q86W56 1/20 0.44
MAPT P10636 6/20 0.43
TSHR P16473 2/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTT P42858 1/20 0.43
POLB P06746 4/20 0.42
TP53 P04637 3/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3253874 1.00 TDP1 (0.52) TDP1LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL3250591 0.96 PARG (0.48) TDP1LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL3254875 0.93 PARG (0.43) TDP1LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL3255447 0.91 TDP1 (0.52) TDP1LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL3249535 0.91 TDP1 (0.51) TDP1LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL3242986 0.90 PARG (0.40) TDP1LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL3251597 0.89 PARG (0.47) TDP1LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL3250743 0.87 KDM4E (0.39) TDP1LMNASMN1; SMN2MAPTHSD17B10
SCHEMBL3247256 0.86 TDP1 (0.53) TDP1LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL3250480 0.86 TDP1 (0.53) TDP1LMNAALDH1A1SMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed