SCHEMBL3253124

SCHEMBL3253124

[C]#Cc1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 3/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
ALDH1A1 P00352 4/20 0.38
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MCL1 Q07820 3/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.36
MAPT P10636 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
ADRA2A P08913 1/20 0.36
AHR P35869 1/20 0.35
CHRNA7 P36544 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9996467 0.84 PDE2A (0.44) PDE2AALDH1A1MEN1TSHRKMT2A
SCHEMBL384969 0.80 AR (0.47) PDE2APTGDR2ALDH1A1HTTSMN1; SMN2
SCHEMBL16951053 0.80 PDE2A (0.41) PDE2APTGDR2ALDH1A1MEN1TSHR
SCHEMBL2651995 0.80 PTGDR2 (0.43) PDE2APTGDR2ALDH1A1MEN1TSHR
SCHEMBL2515789 0.80 PTGDR2 (0.43) PDE2APTGDR2ALDH1A1MEN1TSHR
SCHEMBL29837271 0.80 AR (0.47) PDE2APTGDR2ALDH1A1HTTSMN1; SMN2
SCHEMBL9996392 0.78 CES2 (0.46) PDE2AALDH1A1TSHRHSD17B10
SCHEMBL5545019 0.75 PTGDR2 (0.40) PDE2APTGDR2ALDH1A1MEN1TSHR
SCHEMBL9996732 0.73 AR (0.49)
SCHEMBL980201 0.73 TSHR (0.61) PDE2AALDH1A1MEN1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773330-B1 SUBSTITUTED PYRAZOLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK SHARP & DOHME (US) 2010-05-26 EP disclosed