SCHEMBL3254471

SCHEMBL3254471

COc1ccc2c(c1)CCN(C(=O)CN1C(=O)COc3cc(-c4cc(Cl)cc(Cl)c4)cnc31)C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
GAA P10253 1/20 0.46
MAPK1 P28482 3/20 0.41
MAPT P10636 3/20 0.41
ESR2 Q92731 2/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
POLB P06746 1/20 0.41
NR4A1 P22736 1/20 0.41
APEX1 P27695 1/20 0.41
RECQL P46063 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ESR1 P03372 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
ABCB1 P08183 2/20 0.40
ABHD6 Q9BV23 1/20 0.38
TP53 P04637 1/20 0.38
CA1 P00915 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3241489 0.97 TSHR (0.46) TSHRGAAMAPK1MAPTESR2
SCHEMBL13521687 0.94 GAA (0.39) TSHRGAAMAPK1ALDH1A1TP53
SCHEMBL3241049 0.93 TSHR (0.46) TSHRGAAMAPK1MAPTESR2
SCHEMBL3251960 0.92 TSHR (0.43) TSHRGAAMAPK1MAPTESR2
SCHEMBL3252753 0.91 TSHR (0.44) TSHRGAAMAPK1MAPTESR2
SCHEMBL3251252 0.90 GAA (0.47) TSHRGAAMAPK1ESR2KDM4E
SCHEMBL3248197 0.90 TSHR (0.46) TSHRGAAMAPK1MAPTESR2
SCHEMBL13521136 0.90 TSHR (0.56) TSHRGAAMAPK1MAPTALDH1A1
SCHEMBL3247872 0.89 GAA (0.46) TSHRGAAMAPK1ALDH1A1POLB
SCHEMBL3236789 0.89 GAA (0.55) TSHRGAAMAPK1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010008777-A2 FUSED AZABICYCLIC PYRIDINES LIGAND PHARMACEUTICALS INC. (US) 2010-01-21 WO claimed