SCHEMBL3255505

SCHEMBL3255505

CCOC(=O)Oc1c[nH]c2c(=O)[nH]c3ccc(-c4cccc(CO)c4)cc3c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.39
WEE1 P30291 1/20 0.39
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
DHODH Q02127 1/20 0.36
CSF1R P07333 1/20 0.36
NPC1 O15118 1/20 0.36
CLEC4M Q9H2X3 1/20 0.35
TYMS P04818 1/20 0.35
GABRA1 P14867 2/20 0.35
GABRB2 P47870 2/20 0.35
GABRB1 P18505 1/20 0.35
GABRA3 P34903 1/20 0.35
MAP2K4 P45985 1/20 0.34
HPGD P15428 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3251517 0.90 GRIN2D (0.36) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3245580 0.90 TLR8 (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3252380 0.89 CSF1R (0.43) CHEK1WEE1CSF1RNPC1GABRA1
SCHEMBL3252050 0.89 GAA (0.40) CHEK1WEE1CSF1RNPC1CLEC4M
SCHEMBL3249476 0.88 ICMT (0.37) CHEK1WEE1CSF1RNPC1CLEC4M
SCHEMBL3254793 0.85 HRH2 (0.40) CHEK1WEE1CSF1RNPC1TYMS
SCHEMBL3252205 0.85 TTK (0.42) CHEK1DHODHHPGDALDH1A1KMT2A
SCHEMBL3250925 0.85 NR1H2 (0.38) WEE1CSF1RNPC1CLEC4MTYMS
SCHEMBL3254531 0.85 CLEC4M (0.45) CSF1RNPC1CLEC4MGABRA1GABRB2
SCHEMBL3253850 0.85 SCN9A (0.38) CHEK1WEE1CSF1RNPC1CLEC4M

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed