SCHEMBL3257233

SCHEMBL3257233

Cc1c(C#N)c(Nc2ncnc3c2c2c(n3Cc3ccccc3)CCCC2)n(-c2cccc(Cl)c2)c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
LMNA P02545 3/20 0.38
MAPT P10636 3/20 0.38
NPC1 O15118 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
HTT P42858 3/20 0.38
MITF O75030 1/20 0.38
RAB9A P51151 1/20 0.37
NR2F2 P24468 1/20 0.37
NPSR1 Q6W5P4 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDE1B Q01064 1/20 0.36
SLC2A1 P11166 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3259755 0.89 ALDH1A1 (0.41) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL3262074 0.87 MEN1 (0.47) ALDH1A1MEN1KMT2AMAPTNPC1
SCHEMBL3167119 0.84 ALDH1A1 (0.52) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL3254913 0.80 ABCC1 (0.43) ALDH1A1MEN1KMT2ALMNANPC1
SCHEMBL7497953 0.77 EGFR (0.54) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL3160382 0.77 KMT2A (0.44) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL3259092 0.73 KMT2A (0.64) ALDH1A1MEN1KMT2AMAPTNPC1
SCHEMBL3257449 0.72 CA1 (0.46) MEN1KMT2ANPC1RAB9ASLC2A1
SCHEMBL3171306 0.70 MEN1 (0.54) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL8088056 0.70 EGFR (0.53) ALDH1A1MAPTMKNK1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756110-B1 7H-PYRROLO[2,3-d]PYRIMIDINE DERIVATIVES, AS WELL AS THEIR THERAPEUTICALLY ACCEPTABLE SALTS, PHARMACEUTICAL PREPARATIONS CONTAINING THEM AND PROCESS FOR PRODUCTION THE ACTIVE AGENT SZOLCSANYI JANOS (HU) 2010-03-31 EP disclosed