SCHEMBL3258068

SCHEMBL3258068

O=C(Nc1cc(-c2nc3ccccc3[nH]2)cs1)c1cccc(F)c1.O=C(O)c1c(-c2c[nH]c3ccccc23)csc1Nc1cccc(F)c1.O=C(O)c1c(-c2nc3ccccc3n2C(F)F)csc1Nc1cccc(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.37
MMP2 P08253 2/20 0.36
MMP9 P14780 2/20 0.36
MMP8 P22894 2/20 0.36
MMP13 P45452 2/20 0.36
COMT P21964 1/20 0.36
BACE1 P56817 4/20 0.36
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
MAPT P10636 6/20 0.35
KDM4E B2RXH2 5/20 0.34
POLB P06746 3/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 3/20 0.34
HPGD P15428 3/20 0.34
RECQL P46063 2/20 0.34
LMNA P02545 2/20 0.34
THRB P10828 1/20 0.34
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2179504 0.87 RAB9A (0.45) PDPK1MMP2MMP9MMP8MMP13
SCHEMBL2181427 0.77 MEN1 (0.48) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL2179507 0.75 PDPK1 (0.44) PDPK1MMP2MMP9MMP8MMP13
SCHEMBL7950439 0.74 MEN1 (0.52) BACE1NPC1RAB9AMAPTPOLB
SCHEMBL15241644 0.74 NPC1 (0.62) PDPK1MMP2MMP9MMP8MMP13
SCHEMBL2181392 0.72 RAB9A (0.58) PDPK1MMP2MMP9MMP8MMP13
SCHEMBL3251954 0.72 MTOR (0.48) PDPK1MMP2MMP9MMP8MMP13
SCHEMBL12414216 0.66 FOXO1 (0.61) MMP2MMP9MMP8MMP13COMT
SCHEMBL12830503 0.66 MEN1 (0.42) NPC1RAB9AMAPTKDM4EPOLB
SCHEMBL12434682 0.66 NPC1 (0.57) PDPK1MMP2MMP9MMP8MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025295-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2010-03-04 WO disclosed