SCHEMBL3258236

SCHEMBL3258236

COc1cn(C)c(C2CCN(C(=O)OC(C)(C)C)CC2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
MAPT P10636 1/20 0.47
THRB P10828 1/20 0.47
HTT P42858 2/20 0.46
ALDH1A1 P00352 3/20 0.46
HPGD P15428 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
TSHR P16473 1/20 0.45
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
HSD17B10 Q99714 1/20 0.45
GPR119 Q8TDV5 6/20 0.44
HPGDS O60760 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PDE4B Q07343 1/20 0.42
PTPN2 P17706 1/20 0.42
PTPN1 P18031 1/20 0.42
PTPN6 P29350 1/20 0.42
STS P08842 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16716879 0.86 THRB (0.48) KDM4EMAPTTHRBHTTHPGD
SCHEMBL3262079 0.85 KDM4E (0.49) KDM4EMAPTTHRBHTTHPGD
SCHEMBL16992147 0.82 KDM4E (0.46) KDM4EMAPTTHRBGPR119HPGDS
SCHEMBL22712403 0.76 THRB (0.50) KDM4EMAPTTHRBHTTHPGD
SCHEMBL948563 0.76 GPR119 (0.53) KDM4EMAPTTHRBGPR119HPGDS
SCHEMBL15732488 0.76 P2RY14 (0.51) KDM4EMAPTHTTALDH1A1HPGD
SCHEMBL16434944 0.76 HTT (0.51) KDM4EMAPTTHRBHTTALDH1A1
SCHEMBL31639582 0.75 HTT (0.53) KDM4EMAPTTHRBHTTALDH1A1
SCHEMBL18865690 0.75 KDM4E (0.49) KDM4EMAPTTHRBHTTALDH1A1
SCHEMBL31639499 0.75 GPR119 (0.50) KDM4EMAPTTHRBHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109851610-B Bicyclic aza compounds as muscarinic M1 and/or M4 receptor agonists 赫普泰雅治疗有限公司 2021-09-21 CN disclosed
EP-2150269-A1 NEW CYCLIC PEPTIDE COMPOUNDS Astellas Pharma Inc. (JP) 2010-02-10 EP disclosed
WO-2008139986-A1 NEW CYCLIC PEPTIDE COMPOUNDS ASTELLAS PHARMA INC., (JP) 2008-11-20 WO disclosed