SCHEMBL3259243

SCHEMBL3259243

Brc1ccc2cc3cc4ccccc4cc3cc2c1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.44
HSD17B10 Q99714 6/20 0.44
HIF1A Q16665 2/20 0.44
CYP1B1 Q16678 1/20 0.44
CYP2A6 P11509 5/20 0.43
TDP1 Q9NUW8 3/20 0.41
CYP3A4 P08684 2/20 0.41
ALOX15 P16050 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HBB P68871 1/20 0.41
POLB P06746 1/20 0.38
KDM4E B2RXH2 3/20 0.37
GAA P10253 2/20 0.37
CYP1A2 P05177 5/20 0.36
ERBB2 P04626 1/20 0.36
FYN P06241 1/20 0.36
MAOA P21397 1/20 0.36
ACHE P22303 1/20 0.36
AHR P35869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5010132 1.00 ALDH1A1 (0.44) ALDH1A1HSD17B10HIF1ACYP1B1CYP2A6
SCHEMBL5012382 1.00 ALDH1A1 (0.44) ALDH1A1HSD17B10HIF1ACYP1B1CYP2A6
SCHEMBL5013845 1.00 ALDH1A1 (0.44) ALDH1A1HSD17B10HIF1ACYP1B1CYP2A6
SCHEMBL1004096 0.98 ALDH1A1 (0.46) ALDH1A1HSD17B10HIF1ACYP1B1CYP2A6
SCHEMBL29891613 0.98 ALDH1A1 (0.46) ALDH1A1HSD17B10HIF1ACYP1B1CYP2A6
Anthraquinone SCHEMBL28175362 0.85 CES1 (0.44) ALDH1A1HSD17B10HIF1ACYP1B1CYP3A4
SCHEMBL17967022 0.83 CYP1A2 (0.42) ALDH1A1HSD17B10HIF1ACYP1B1CYP2A6
SCHEMBL25966 0.78 ALDH1A1 (0.68) ALDH1A1HSD17B10HIF1ACYP1B1CYP2A6
SCHEMBL190685 0.78 ALDH1A1 (0.68) ALDH1A1HSD17B10HIF1ACYP1B1CYP2A6
SCHEMBL15063036 0.78 ALDH1A1 (0.68) ALDH1A1HSD17B10HIF1ACYP1B1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112694388-A Naphthacene derivative and preparation method and application thereof 中国科学院化学研究所 2021-04-23 CN disclosed
US-7651746-B2 Halogenated bisdiarylaminopolycyclic aromatic compounds and polymers thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-01-26 US disclosed
CN-100482634-C Organic electroluminescent device IDEMITSU PETROCHEMICAL CO (JP) 2009-04-29 CN disclosed
US-20070126345-A1 Halogenated bisdiarylaminopolycylic aromatic compounds and polymers thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-06-07 US disclosed
CN-1721499-A Organic electroluminescent device IDEMITSU KOSAN CO (JP) 2006-01-18 CN disclosed
CN-1219747-C Organic electroluminescent device IDEMITSU KOSAN CO (JP) 2005-09-21 CN disclosed
WO-2005049546-A1 HALOGENATED BISDIARYLAMINOPOLYCYLIC AROMATIC COMPOUNDS AND POLYMERS THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2005-06-02 WO disclosed
CN-1292022-A Organic electroluminescent device IDEMITSU KOSAN CO (JP) 2001-04-18 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070126345-A1 Halogenated bisdiarylaminopolycylic aromatic compounds and polymers thereof AHR, AADAC, ARNT ALDH1A1 667/4885HSD17B10 951/4885HIF1A 3596/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.