SCHEMBL3260890

SCHEMBL3260890

N=C(NC(=O)O)N1CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
F2 P00734 1/20 0.41
GAA P10253 1/20 0.39
HPGD P15428 4/20 0.37
POLB P06746 1/20 0.37
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MMP9 P14780 1/20 0.37
HTT P42858 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
CA2 P00918 1/20 0.35
CHKA P35790 1/20 0.35
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15588799 0.83 F2 (0.50) ALDH1A1F2GAAHPGDPOLB
SCHEMBL15588798 0.83 F2 (0.50) ALDH1A1F2GAAHPGDPOLB
Hydrochloric Acid SCHEMBL16766200 0.80 F2 (0.48) ALDH1A1F2GAAHPGDPOLB
Hydrochloric Acid SCHEMBL16766683 0.80 F2 (0.48) ALDH1A1F2GAAHPGDPOLB
SCHEMBL17336983 0.80 F2 (0.50) ALDH1A1F2GAAHPGDPOLB
SCHEMBL15588635 0.80 F2 (0.46) ALDH1A1F2HPGDPOLBHTT
SCHEMBL17186605 0.79 GAA (0.44) ALDH1A1F2GAAPOLBHTT
SCHEMBL7108628 0.78 CA2 (0.43) HPGDPOLBCA2CHKAHSD11B1
Acetic Acid SCHEMBL17417178 0.78 F2 (0.43) ALDH1A1F2GAAHPGDPOLB
Hydrochloric Acid SCHEMBL15560657 0.78 F2 (0.43) ALDH1A1F2HPGDPOLBCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7649000-B2 (2'S,2''R)-4-(2'-(2''-amino-3''-(4'''-ethoxyphenyl)propanoylamino)-3'-phenylpropanoyl-amino)piperidine- 1-carboxamidine; inflammatory bowel disease, arthritis, inflammation, septic shock, hypotension, cancer, adult respiratory distress syndrome, disseminated intravascular coagulation VANTIA LIMITED (GB) 2010-01-19 US disclosed
EP-1483284-B1 SELECTIVE DIPEPTIDE INHIBITORS OF KALLIKREIN FERRING BV (NL) 2006-07-19 EP disclosed
US-20060052313-A1 Selective dipeptide inhibitors of kallikrein FERRING B.V 2006-03-09 US disclosed
EP-1483284-A2 SELECTIVE DIPEPTIDE INHIBITORS OF KALLIKREIN Ferring BV (NL) 2004-12-08 EP disclosed
WO-2003076458-A2 SELECTIVE DIPEPTIDE INHIBITORS OF KALLIKREIN FERRING BV (NL) 2003-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052313-A1 Selective dipeptide inhibitors of kallikrein BDKRB2, BDKRB1, KLKB1 ALDH1A1 3712/4885F2 108/4885GAA 3328/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.