SCHEMBL3262109

SCHEMBL3262109

COC(=O)N1CCc2ccccc2C(c2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAPK1 P28482 2/20 0.46
KIF11 P52732 1/20 0.46
MAPK14 Q16539 1/20 0.46
BRD4 O60885 1/20 0.44
HAO1 Q9UJM8 1/20 0.44
HDAC8 Q9BY41 2/20 0.43
PRCP P42785 1/20 0.43
CHRM3 P20309 2/20 0.42
CACNA1F O60840 1/20 0.42
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM5 P08912 1/20 0.42
CHRM1 P11229 1/20 0.42
KCNE1 P15382 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6097273 0.79 NOTUM (0.58) ALDH1A1MAPTTSHRMAPK1MEN1
SCHEMBL3260780 0.76 PRCP (0.57) KDM4EMAPTMAPK1PRCPSIGMAR1
SCHEMBL31073550 0.76 KCNH2 (0.56) ALDH1A1LMNAL3MBTL1MAPK1BRD4
SCHEMBL3260783 0.76 PRCP (0.57) KDM4EMAPTMAPK1PRCPSIGMAR1
SCHEMBL13589929 0.75 CHRM3 (0.62) HDAC8PRCPCHRM3CACNA1FCHRM2
SCHEMBL1566898 0.75 CHRM3 (0.62) HDAC8PRCPCHRM3CACNA1FCHRM2
Bicarbonate SCHEMBL376797 0.74 SIGMAR1 (0.55) MAPK1MAPK14HAO1SIGMAR1MEN1
Butanedione SCHEMBL17273471 0.73 SIGMAR1 (0.55) TSHRMAPK1MAPK14HAO1GID4
SCHEMBL464005 0.71 NOTUM (0.67) ALDH1A1MAPTMEN1CYP3A4CYP2C19
SCHEMBL30056523 0.71 NOTUM (0.67) ALDH1A1MAPTMEN1CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010012812-A1 BENZAZEPINES AND BENZAZOCINES AS SIGMA-RECEPTOR LIGANDES Westfälische Wilhelms Universität Münster (DE) 2010-02-04 WO disclosed