SCHEMBL3262157

SCHEMBL3262157

Cc1ccccc1-n1nc(C)c(-c2ccc3nc(N)nn3c2)c1[NH]

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
PIK3CG P48736 7/20 0.38
PIK3CD O00329 6/20 0.38
PIK3CA P42336 3/20 0.38
PIK3CB P42338 2/20 0.38
OPRM1 P35372 1/20 0.35
LRRK2 Q5S007 3/20 0.35
JAK2 O60674 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MAP4K4 O95819 1/20 0.32
PAK4 O96013 1/20 0.32
CSF1R P07333 1/20 0.32
RET P07949 1/20 0.32
GRK5 P34947 1/20 0.32
MAPK8 P45983 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3262160 0.88 HTT (0.45) ALDH1A1MAPTHTTKMT2APIK3CG
SCHEMBL7937768 0.75 ADORA1 (0.53) LRRK2ADORA1
SCHEMBL614711 0.68 RET (0.61) ALDH1A1PIK3CGPIK3CDPIK3CAPIK3CB
SCHEMBL2186588 0.66 PIK3CG (0.60) PIK3CGPIK3CDPIK3CAPIK3CBLRRK2
SCHEMBL936441 0.65 PIK3CG (0.51) ALDH1A1PIK3CGPIK3CDPIK3CAPIK3CB
SCHEMBL6181854 0.64 HTT (0.47) ALDH1A1MAPTHTTKMT2AOPRM1
SCHEMBL1933137 0.64 PIK3CG (0.52) ALDH1A1MAPTKMT2APIK3CGPIK3CD
SCHEMBL3974032 0.64 SMN1; SMN2 (0.54) ALDH1A1MAPTHTTKMT2ANPC1
SCHEMBL10044580 0.63 PIK3CG (0.44) ALDH1A1KMT2APIK3CGPIK3CDPIK3CA
SCHEMBL936292 0.63 PIK3CD (0.61) ALDH1A1PIK3CGPIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010020363-A1 SUBSTITUTED 5-AMINOPYRAZOLES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-25 WO disclosed