SCHEMBL6181854

SCHEMBL6181854

Cc1ccccc1-n1nc(N)nc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 5/20 0.46
MAPT P10636 2/20 0.46
TSHR P16473 2/20 0.41
MAPK14 Q16539 1/20 0.40
HCAR1 Q9BXC0 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
TP53 P04637 2/20 0.40
OPRM1 P35372 1/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
FLT3 P36888 2/20 0.37
GSK3B P49841 1/20 0.37
LMNA P02545 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HIF1A Q16665 1/20 0.37
PI4KA P42356 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11201816 0.79 FLT3 (0.49) ALDH1A1TSHRMAPK14HCAR1TP53
SCHEMBL4884376 0.78 FLT3 (0.48) KMT2AALDH1A1MAPK14HCAR1TDP1
SCHEMBL5354248 0.77 FLT3 (0.48) KMT2AALDH1A1MAPK14ADORA3ADORA2A
SCHEMBL8942018 0.72 TSHR (0.58) KMT2AALDH1A1MAPTTSHRMAPK1
SCHEMBL16458811 0.71 NUDT1 (0.46) MAPK1FLT3NUDT1
SCHEMBL1143383 0.70 CYP1A2 (0.62) HTTKMT2AALDH1A1MAPTTSHR
SCHEMBL28455262 0.70 ALDH1A1 (0.62) HTTKMT2AALDH1A1MAPTTSHR
SCHEMBL30258577 0.69 HCAR1 (0.43) HTTKMT2AALDH1A1HCAR1LMNA
Hydrochloric Acid SCHEMBL11473767 0.69 CYP1A2 (0.61) HTTKMT2AALDH1A1MAPTTSHR
SCHEMBL1816971 0.68 POLB (0.55) HTTKMT2AALDH1A1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104428289-B As the triazole compounds of antivirotic 弗·哈夫曼-拉罗切有限公司 2017-06-23 CN claimed
EP-1126843-A4 COMPOUNDS DERIVED FROM AN AMINE NUCLEUS THAT ARE INHIBITORS OF IMPDH ENZYME BRISTOL MYERS SQUIBB CO (US) 2005-06-15 EP disclosed
EP-1126843-A1 COMPOUNDS DERIVED FROM AN AMINE NUCLEUS THAT ARE INHIBITORS OF IMPDH ENZYME BRISTOL-MYERS SQUIBB COMPANY (US) 2001-08-29 EP disclosed
WO-2000025780-A1 COMPOUNDS DERIVED FROM AN AMINE NUCLEUS THAT ARE INHIBITORS OF IMPDH ENZYME BRISTOL-MYERS SQUIBB COMPANY (US) 2000-05-11 WO disclosed