SCHEMBL3262865

SCHEMBL3262865

Nc1nc2cccc(N3CCNCC3)n2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 4/20 0.45
EGLN2 Q96KS0 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
HRH4 Q9H3N8 3/20 0.41
JAK1 P23458 2/20 0.40
HTR3E A5X5Y0 2/20 0.40
HTR3B O95264 2/20 0.40
HTR3A P46098 2/20 0.40
HTR3D Q70Z44 2/20 0.40
HTR3C Q8WXA8 2/20 0.40
ALDH1A1 P00352 1/20 0.40
ABCB1 P08183 1/20 0.39
NCF1 P14598 2/20 0.38
HTR2A P28223 2/20 0.37
ADRB1 P08588 2/20 0.37
CYP1A2 P05177 1/20 0.37
HTR1A P08908 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2250437 0.86 NUDT1 (0.57) NUDT1EGLN2JAK1ALDH1A1CYP1A2
SCHEMBL2254109 0.84 NUDT1 (0.60) NUDT1EGLN2JAK1ALDH1A1CYP1A2
SCHEMBL2253273 0.84 NUDT1 (0.60) NUDT1EGLN2JAK1ALDH1A1CYP1A2
SCHEMBL2252271 0.83 NUDT1 (0.46) NUDT1EGLN2JAK1ALDH1A1NCF1
SCHEMBL3261461 0.81 NUDT1 (0.44) NUDT1EGLN2HRH3HRH4JAK1
SCHEMBL3591147 0.78 NUDT1 (0.59) NUDT1EGLN2JAK1HTR3EHTR3B
SCHEMBL3262068 0.77 NUDT1 (0.46) NUDT1EGLN2HRH3HRH4JAK1
SCHEMBL3216262 0.76 JAK1 (0.44) NUDT1EGLN2JAK1ALDH1A1MTOR
SCHEMBL4499154 0.72 PRKCI (0.45) HRH3HRH4HTR3AABCB1ADRB1
SCHEMBL18077197 0.72 EGLN2 (0.62) EGLN2ALDH1A1HTR2AADRB1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010010187-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE AND INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2010-01-28 WO disclosed