SCHEMBL3263341

SCHEMBL3263341

CNC(=O)c1c(C)oc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 6/20 0.58
EYA3 Q99504 3/20 0.58
CYP2C9 P11712 3/20 0.50
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
GAA P10253 1/20 0.44
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
HPGD P15428 1/20 0.43
HIF1A Q16665 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KDM7A Q6ZMT4 1/20 0.43
EGFR P00533 1/20 0.43
SRC P12931 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30753455 0.82 CYP2C19 (0.54) CYP2C19EYA3CYP2C9ALDH1A1KDM4E
SCHEMBL30753472 0.82 CYP2C19 (0.54) CYP2C19EYA3CYP2C9KDM4ENPC1
SCHEMBL9657351 0.80 CYP2C19 (0.63) CYP2C19EYA3CYP2C9NPC1RAB9A
SCHEMBL1398779 0.80 CYP2C19 (0.63) CYP2C19EYA3CYP2C9ALDH1A1KDM4E
SCHEMBL18018241 0.79 CYP2C19 (0.61) CYP2C19EYA3CYP2C9ALDH1A1KDM4E
SCHEMBL5241666 0.79 GAA (0.52) CYP2C19EYA3CYP2C9ALDH1A1KDM4E
SCHEMBL26335570 0.79 CA12 (0.56) CYP2C19CYP2C9ALDH1A1KDM4EHPGD
SCHEMBL944525 0.79 GAA (0.52) CYP2C19EYA3CYP2C9ALDH1A1KDM4E
SCHEMBL4670295 0.79 CYP2C19 (0.61) CYP2C19EYA3CYP2C9ALDH1A1KDM4E
SCHEMBL20441188 0.79 CYP2C19 (0.61) CYP2C19EYA3CYP2C9KDM4ETHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260022125-A1 PYRROLOPYRIDAZINE VEGFR INHIBITORS MERCK SHARP & DOHME LLC (US) 2026-01-22 US claimed
CN-117285518-A Quinazoline derivative containing benzofuran structure and application thereof 华侨大学 2023-12-26 CN claimed
US-20260022125-A1 PYRROLOPYRIDAZINE VEGFR INHIBITORS MERCK SHARP & DOHME LLC (US) 2026-01-22 US disclosed
CN-120051468-A Hydrate of VEGFR inhibitor, crystal form thereof and preparation method thereof 成都苑东生物制药股份有限公司 2025-05-27 CN disclosed
CN-120051468-A Hydrate of VEGFR inhibitor, crystal form thereof and preparation method thereof 成都苑东生物制药股份有限公司 2025-05-27 CN disclosed
CN-120025319-A New crystal form of quinazoline compound 南京正大天晴制药有限公司 2025-05-23 CN disclosed
CN-120025320-A Quinazoline hydrate of compound 南京正大天晴制药有限公司 2025-05-23 CN disclosed
CN-117285518-A Quinazoline derivative containing benzofuran structure and application thereof 华侨大学 2023-12-26 CN disclosed
CN-115003332-A Application of anti-PD-1 antibody and furoquintinib combination in preparation of medicine for treating cancer 嘉和生物药业有限公司 2022-09-02 CN disclosed
CN-113200966-B Furosetinib derivative, pharmaceutical composition and application 深圳大学 2022-07-22 CN disclosed
WO-2010025138-A2 PYRIMIDINE COMPOUNDS HUTCHISON MEDIPHARMA ENTERPRISES LIMITED (BS) 2010-03-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260022125-A1 PYRROLOPYRIDAZINE VEGFR INHIBITORS FLT1, KDR, FLT4 CYP2C19 166/4885EYA3 3188/4885CYP2C9 159/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.