SCHEMBL3264111

SCHEMBL3264111

CCOC(=O)c1ccc(-c2cccc3nc(N)nn23)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 6/20 0.60
NUDT1 P36639 3/20 0.57
EGLN2 Q96KS0 1/20 0.53
JAK3 P52333 1/20 0.50
LMNA P02545 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
MAOA P21397 1/20 0.48
PARP1 P09874 1/20 0.44
RARA P10276 1/20 0.43
RARB P10826 1/20 0.43
RARG P13631 1/20 0.43
JAK2 O60674 1/20 0.43
PDE4A P27815 1/20 0.43
ALDH1A1 P00352 2/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
PKM P14618 1/20 0.42
RAB9A P51151 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3264207 0.80 NUDT1 (0.72) JAK1NUDT1EGLN2JAK3JAK2
SCHEMBL22499606 0.79 NUDT1 (0.73) JAK1NUDT1EGLN2JAK3LMNA
SCHEMBL3657387 0.77 JAK2 (0.61) JAK1JAK3JAK2RAB9A
SCHEMBL13072986 0.77 JAK2 (0.76) JAK1JAK3JAK2RAB9A
SCHEMBL3601961 0.75 NUDT1 (0.78) JAK1NUDT1EGLN2JAK3JAK2
SCHEMBL3090231 0.75 JAK1 (1.00) JAK1NUDT1EGLN2JAK3JAK2
SCHEMBL3588844 0.73 NUDT1 (0.57) JAK1NUDT1EGLN2JAK3JAK2
SCHEMBL2250300 0.73 NUDT1 (0.73) JAK1NUDT1EGLN2JAK3JAK2
SCHEMBL2363033 0.73 NUDT1 (0.73) JAK1NUDT1EGLN2JAK3LMNA
SCHEMBL2634912 0.73 JAK3 (0.65) JAK1NUDT1EGLN2JAK3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010010189-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE AND INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2010-01-28 WO disclosed
WO-2010010189-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE AND INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2010-01-28 WO disclosed