SCHEMBL3264199

SCHEMBL3264199

COc1cc(C(F)(F)F)ccc1C(=O)NC(c1ccccc1)C1(N2CCCC2)CCC1.CSc1cc(C(F)(F)F)ccc1C(=O)NC(c1ccccc1)C1(N2CCCC2)CCC1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 14/20 0.47
MTTP P55157 5/20 0.46
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
SLC6A5 Q9Y345 1/20 0.45
AVPR2 P30518 1/20 0.39
GPR27 Q9NS67 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1349364 0.93 SLC6A9 (0.53) SLC6A9MTTPAVPR2GPR27
SCHEMBL1347772 0.93 SLC6A9 (0.53) SLC6A9MTTPCYP2D6CYP2C19SLC6A5
SCHEMBL1349456 0.93 SLC6A9 (0.52) SLC6A9MTTPCYP2D6CYP2C19SLC6A5
SCHEMBL1350169 0.91 SLC6A9 (0.54) SLC6A9MTTPCYP2D6CYP2C19SLC6A5
SCHEMBL1349513 0.88 SLC6A9 (0.56) SLC6A9CYP2D6CYP2C19SLC6A5
SCHEMBL1349692 0.87 SLC6A9 (0.55) SLC6A9CYP2D6CYP2C19SLC6A5
SCHEMBL1348599 0.87 SLC6A9 (0.50) SLC6A9MTTP
SCHEMBL1350069 0.86 SLC6A9 (0.46) SLC6A9
SCHEMBL1349875 0.85 SLC6A9 (0.46) SLC6A9CYP2C19
SCHEMBL1348719 0.85 SLC6A9 (0.57) SLC6A9CYP2D6CYP2C19SLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010020548-A1 GLYT1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-02-25 WO disclosed