SCHEMBL3264297

SCHEMBL3264297

O=C(Nc1ccccc1)c1cnns1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 1/20 0.65
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
KDM4E B2RXH2 1/20 0.50
PPARG P37231 1/20 0.49
NCOA2 Q15596 1/20 0.49
NCOA1 Q15788 1/20 0.49
NCOA3 Q9Y6Q9 1/20 0.49
PTPN1 P18031 3/20 0.48
P4HTM Q9NXG6 1/20 0.47
POLB P06746 1/20 0.47
EGFR P00533 2/20 0.47
LCK P06239 1/20 0.47
HTT P42858 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
TP53 P04637 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15074544 0.83 RAB9A (0.54) RPS6KA3NPC1RAB9AALDH1A1KDM4E
SCHEMBL15076235 0.83 RPS6KA3 (0.57) RPS6KA3NPC1RAB9AALDH1A1LMNA
SCHEMBL2732134 0.83 RPS6KA3 (0.54) RPS6KA3NPC1RAB9AALDH1A1LMNA
Thidiazuron SCHEMBL1808496 0.75 SMN1; SMN2 (0.57) NPC1RAB9AALDH1A1LMNAKDM4E
Thidiazuron SCHEMBL121077 0.75 SMN1; SMN2 (0.57) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL11925387 0.73 PTPN1 (0.59) NPC1RAB9AALDH1A1LMNAKDM4E
Thidiazuron SCHEMBL15553871 0.73 SMN1; SMN2 (0.55) NPC1RAB9AALDH1A1LMNAKDM4E
Thidiazuron SCHEMBL20723866 0.73 SMN1; SMN2 (0.55) NPC1RAB9AALDH1A1LMNAKDM4E
SCHEMBL27795863 0.73 RPS6KA3 (0.49) RPS6KA3
SCHEMBL892780 0.72 KMT2A (0.71) NPC1RAB9AALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025870-A1 SYNERGISTIC COMBINATIONS OF THIADIAZOL CARBONIC ACID DERIVATIVES BAYER CROPSCIENCE AG (DE) 2010-03-11 WO disclosed
EP-1896417-A1 LINEAR UREA MIMICS ANTAGONISTS OF P2Y1 RECEPTOR USEFUL IN THE TREATMENT OF THROMBOTIC CONDITIONS Brystol-Myers Squibb Company (US) 2008-03-12 EP disclosed
WO-2007002584-A1 LINEAR UREA MIMICS ANTAGONISTS OF P2Y1 RECEPTOR USEFUL IN THE TREATMENT OF THROMBOTIC CONDITIONS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed