SCHEMBL3264766

SCHEMBL3264766

COC(=O)c1ccccc1-c1ccc(CNC(=O)C2CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 6/20 0.53
SLC6A3 Q01959 4/20 0.53
SLC6A4 P31645 3/20 0.53
ALDH1A1 P00352 3/20 0.51
HPGD P15428 2/20 0.51
USP2 O75604 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.49
NPC1 O15118 1/20 0.48
PKM P14618 1/20 0.48
RAB9A P51151 1/20 0.48
SLC6A2 P23975 1/20 0.48
SCN9A Q15858 2/20 0.47
CHRNB2 P17787 1/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA4 P43681 1/20 0.47
LTB4R2 Q9NPC1 1/20 0.46
KDM4E B2RXH2 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3109493 0.80 BDKRB1 (0.61) BDKRB1SLC6A3SLC6A4ALDH1A1SLC6A2
SCHEMBL2782748 0.80 CHRNB2 (0.59) BDKRB1SLC6A3SLC6A4SMN1; SMN2NPC1
SCHEMBL5782374 0.79 BDKRB1 (0.60) BDKRB1SLC6A3SLC6A4ALDH1A1SLC6A2
SCHEMBL5061628 0.79 SLC6A3 (0.61) BDKRB1SLC6A3SLC6A4ALDH1A1SMN1; SMN2
SCHEMBL5924515 0.79 SLC6A3 (0.55) BDKRB1SLC6A3SLC6A4ALDH1A1SLC6A2
SCHEMBL5783245 0.78 BDKRB1 (0.68) BDKRB1SLC6A3SLC6A4ALDH1A1SLC6A2
SCHEMBL29979869 0.78 SLC6A3 (0.69) BDKRB1SLC6A3SLC6A4SLC6A2LTB4R2
SCHEMBL3112718 0.78 SLC6A3 (0.69) BDKRB1SLC6A3SLC6A4SLC6A2LTB4R2
SCHEMBL14326964 0.78 SLC6A3 (0.69) BDKRB1SLC6A3SLC6A4SLC6A2LTB4R2
SCHEMBL8872163 0.78 BDKRB1 (0.70) BDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1706372-B1 ALPHA-HYDROXY AMIDES AS BRADYKININ ANTAGONISTS OR INVERSE AGONISTS MERCK SHARP & DOHME (US) 2010-05-19 EP disclosed