SCHEMBL3265628

SCHEMBL3265628

COc1cc2nc(C)nc(N)c2cc1OC

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 5/20 0.61
KMT2A Q03164 2/20 0.61
LMNA P02545 1/20 0.61
GLA P06280 1/20 0.61
GAA P10253 1/20 0.61
SMARCA2 P51531 1/20 0.61
PDE4A P27815 1/20 0.54
PDE4D Q08499 1/20 0.54
MAPT P10636 6/20 0.54
TP53 P04637 5/20 0.54
BLM P54132 2/20 0.54
RAD52 P43351 2/20 0.54
MEN1 O00255 1/20 0.54
MITF O75030 1/20 0.54
KDM4E B2RXH2 1/20 0.52
APAF1 O14727 1/20 0.52
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
UBE2N P61088 1/20 0.52
ABCB1 P08183 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27253863 0.89 DHFR (0.50) POLBKMT2ALMNAGLAGAA
SCHEMBL24355432 0.87 PDPK1 (0.57) POLBKMT2ALMNAGLAGAA
SCHEMBL29756065 0.87 PDPK1 (0.57) POLBKMT2ALMNAGLAGAA
SCHEMBL29361482 0.83 POLB (0.63) POLBKMT2ALMNAGLAGAA
SCHEMBL879558 0.83 POLB (0.63) POLBKMT2ALMNAGLAGAA
SCHEMBL13335780 0.81 PDE4A (0.57) POLBKMT2ALMNAGLAGAA
SCHEMBL24355108 0.80 PDE4A (0.45) PDE4APDE4D
SCHEMBL26069641 0.80 POLB (0.49) POLBKMT2ALMNAGLAGAA
SCHEMBL11404500 0.80 POLB (0.59) POLBKMT2ALMNAGLAGAA
SCHEMBL29642054 0.80 POLB (0.59) POLBKMT2ALMNAGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3601267-A1 2-METHYL-QUINAZOLINES Bayer Pharma Aktiengesellschaft (DE) 2020-02-05 EP claimed
WO-2018172250-A1 2-METHYL-QUINAZOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-09-27 WO claimed
US-20240084305-A1 MODULATORS OF CELL PROLIFERATION AND USES THEREOF KUMQUAT BIOSCIENCES INC. 2024-03-14 US disclosed
US-20240083857-A1 2-Methyl-Quinazolines Bayer Pharma AG (DE) 2024-03-14 US disclosed
US-20230322803-A1 SUBSTITUTED OXOISOINDOLINE COMPOUNDS FOR THE TREATMENT OF CANCER BRISTOL MYERS SQUIBB CO (US) 2023-10-12 US disclosed
US-20230322803-A1 SUBSTITUTED OXOISOINDOLINE COMPOUNDS FOR THE TREATMENT OF CANCER BRISTOL MYERS SQUIBB CO (US) 2023-10-12 US disclosed
EP-4225383-A1 MODULATORS OF CELL PROLIFERATION AND USES THEREOF Kumquat Biosciences Inc. (US) 2023-08-16 EP disclosed
US-20220274979-A1 2-METHYL-AZA-QUINAZOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2022-09-01 US disclosed
WO-2022076917-A1 MODULATORS OF CELL PROLIFERATION AND USES THEREOF KUMQUAT BIOSCIENCES INC. (US) 2022-04-14 WO disclosed
WO-2021194914-A1 SUBSTITUTED OXOISOINDOLINE COMPOUNDS FOR THE TREATMENT OF CANCER BRISTOL-MYERS SQUIBB COMPANY (US) 2021-09-30 WO disclosed
WO-2021076617-A1 BROAD SPECTRUM ANTI-CANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-04-22 WO disclosed
US-8034818-B2 Therapeutic uses of derivatives of piperidinyl- and piperazinyl-alkyl carbamates SANOFI-AVENTIS (FR) 2011-10-11 US disclosed
US-8034818-B2 Therapeutic uses of derivatives of piperidinyl- and piperazinyl-alkyl carbamates SANOFI-AVENTIS (FR) 2011-10-11 US disclosed
US-7902373-B2 asthma; for treating prostaglandin D2 mediated diseases; e.g. 6-(3-fluorophenyl)-N-[1-(1-methyl-1H-tetrazol-5-yl)piperidin-4-yl]nicotinamide PFIZER INC (US) 2011-03-08 US disclosed
WO-2009016387-A2 PROCESS FOR THE PREPARATION OF ALFUZOSIN HYDROCHLORIDE CIPLA LIMITED (IN) 2009-02-05 WO disclosed
WO-2008104869-A1 NICOTINAMIDE DERIVATIVES AS INHIBITORS OF H-PGDS AND THEIR USE FOR TREATING PROSTAGLANDIN D2 MEDIATED DISEASES PFIZER PRODUCTS INC. (US) 2008-09-04 WO disclosed
WO-2008075172-A2 NICOTINAMIDE DERIVATIVES AS INHIBITORS OF H-PGDS AND THEIR USE FOR TREATING PROSTAGLANDIN D2 MEDIATED DISEASES PFIZER PRODUCTS INC. (US) 2008-06-26 WO disclosed
US-20080146569-A1 Nicotinamide Derivatives PFIZER INC. 2008-06-19 US disclosed
US-7214798-B2 Derivatives of piperidinyl-and piperazinyl-alkyl carbamates, preparation methods thereof and application of same in therapeutics SANOFI-AVENTIS (FR) 2007-05-08 US disclosed
US-7214798-B2 Derivatives of piperidinyl-and piperazinyl-alkyl carbamates, preparation methods thereof and application of same in therapeutics SANOFI-AVENTIS (FR) 2007-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240083857-A1 2-Methyl-Quinazolines NRAS, KRAS, KSR2 POLB 2591/4885KMT2A 834/4885LMNA 3538/4885
US-20230322803-A1 SUBSTITUTED OXOISOINDOLINE COMPOUNDS FOR THE TREATMENT OF CANCER DDX21, HRAS, RPL17 POLB 719/4885KMT2A 1071/4885LMNA 1074/4885
US-20240084305-A1 MODULATORS OF CELL PROLIFERATION AND USES THEREOF MKI67, MYC, CCNK POLB 1167/4885KMT2A 3192/4885LMNA 2637/4885
US-20220274979-A1 2-METHYL-AZA-QUINAZOLINES AZI2, DNMT1, TPMT POLB 191/4885KMT2A 92/4885LMNA 742/4885
US-20080146569-A1 Nicotinamide Derivatives NNT, NAMPT, NADK POLB 2232/4885KMT2A 2987/4885LMNA 1093/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.