SCHEMBL326586

SCHEMBL326586

O=C=Nc1c(Cl)cccc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.56
GABRB2 P47870 2/20 0.56
TDP1 Q9NUW8 2/20 0.45
MAPK1 P28482 1/20 0.45
CYP3A4 P08684 2/20 0.43
CYP1A2 P05177 2/20 0.38
CYP2A6 P11509 2/20 0.38
ALDH1A1 P00352 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TSHR P16473 4/20 0.36
LMNA P02545 1/20 0.36
HSP90AA1 P07900 1/20 0.35
MAPT P10636 1/20 0.35
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
AKR1B1 P15121 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3635498 0.89 GABRA1 (0.50) GABRA1GABRB2TDP1MAPK1CYP3A4
SCHEMBL462306 0.87 CYP3A4 (0.52) GABRA1GABRB2TDP1MAPK1CYP3A4
SCHEMBL1064753 0.85 GABRA1 (0.47) GABRA1GABRB2TDP1MAPK1CYP3A4
SCHEMBL29648809 0.85 GABRA1 (0.47) GABRA1GABRB2TDP1MAPK1CYP3A4
SCHEMBL30390691 0.85 GABRA1 (0.52) GABRA1GABRB2TDP1MAPK1CYP3A4
SCHEMBL1950281 0.85 GABRA1 (0.47) GABRA1GABRB2TDP1MAPK1CYP3A4
SCHEMBL160980 0.85 GABRA1 (0.52) GABRA1GABRB2TDP1MAPK1CYP3A4
SCHEMBL10615737 0.83 GABRA1 (0.78) GABRA1GABRB2TDP1MAPK1CYP3A4
SCHEMBL10882070 0.83 GABRA1 (0.60) GABRA1GABRB2TDP1MAPK1CYP3A4
SCHEMBL11509303 0.83 GABRA1 (0.60) GABRA1GABRB2TDP1MAPK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 690 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103304446-B Derivatization method of optically active phenylacetylene compound UNIV HARBIN ENG 2015-02-25 CN claimed
EP-1377589-B1 OXAZOLYL-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS PHARMACIA ITALIA SPA (IT) 2005-09-07 EP claimed
US-5134189-A Isocyanate, Imino Compound, Polymeric Binder MITSUBISHI PAPER MILLS LIMITED (JP) 1992-07-28 US claimed
JP-59135188-A None JP disclosed
JP-2107477-A None JP disclosed
JP-59135187-A None JP disclosed
JP-60262686-A None JP disclosed
JP-5338356-A None JP disclosed
JP-3199085-A None JP disclosed
JP-3199086-A None JP disclosed
JP-7108759-A None JP disclosed
US-4239768-A GASTROINTESTINAL DISORDERS MCNEILAB, INC. (US) 1980-12-16 US disclosed
US-4229462-A N-ARYL-N'-(2-IMIDAZOLIDINYLIDENE)UREA MCNEILAB, INC. (US) 1980-10-21 US disclosed
US-4174398-A Combating fungi with 1-alkyl-1-(1,3,4-thiadiazol-2-yl)-3-phenyl-ureas BAYER AKTIENGESELLSCHAFT (DE) 1979-11-13 US disclosed
US-4150158-A Oxadiazindione derivatives useful as insecticides IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1979-04-17 US disclosed
US-4051239-A METHOD OF USE AND PROCESS FOR PREPARING PHOSPHOROIMINOBENZOYLUREA INSECTICIDES STAUFFER CHEMICAL COMPANY (US) 1977-09-27 US disclosed
US-4046909-A Pyrrolidylidene, piperidylidene and hexahydroazepinylidene ureas as CNS depressants MCNEIL LABORATORIES, INCORPORATED (US) 1977-09-06 US disclosed
US-4025517-A 4-Oxo-2-hexahydropyrimidinylidene ureas MCNEIL LABORATORIES, INCORPORATED (US) 1977-05-24 US disclosed
US-3998958-A Pyrrolidylidene, piperidylidene and hexahydroazepinylidene ureas as CNS depressants MCNEIL LABORATORIES, INCORPORATED (US) 1976-12-21 US disclosed
US-3983135-A 4-Oxo-2-imidazolidinylidene ureas MCNEIL LABORATORIES, INCORPORATED (US) 1976-09-28 US disclosed