SCHEMBL3269489

SCHEMBL3269489

NS(=O)(=O)c1ccccc1-c1cccc2nccnc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 7/20 0.50
CA2 P00918 7/20 0.50
CA9 Q16790 5/20 0.50
MAPK1 P28482 1/20 0.50
ALOX5AP P20292 3/20 0.42
FEN1 P39748 3/20 0.42
CA12 O43570 3/20 0.41
FTO Q9C0B1 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
CA4 P22748 2/20 0.39
CA6 P23280 2/20 0.39
CYP2C9 P11712 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18007621 0.84 CA1 (0.62) CA1CA2CA9MAPK1CA12
SCHEMBL3256397 0.81 CA1 (0.73) CA1CA2CA9MAPK1CA12
SCHEMBL18343901 0.79 CA1 (0.61) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL3069598 0.78 KDM4E (0.58) KDM4EMEN1USP2ALDH1A1POLB
SCHEMBL1080972 0.76 CA2 (0.61) CA1CA2CA9ALOX5APFEN1
SCHEMBL28771451 0.75 CA1 (0.53) CA1CA2CA9MAPK1CA12
SCHEMBL8347239 0.74 CA2 (0.58) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL17215298 0.74 CCNB2 (0.47) KDM4EMEN1USP2ALDH1A1POLB
SCHEMBL29434853 0.74 CCNB2 (0.47) KDM4EMEN1USP2ALDH1A1POLB
SCHEMBL8697131 0.73 CA1 (0.47) CA1CA2CA9MAPK1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675526-A1 NOVEL SULFONAMINOQUINOLINE HEPCIDIN ANTAGONISTS Vifor (International) AG (CH) 2013-12-25 EP disclosed
WO-2012110603-A1 NOVEL SULFONAMINOQUINOLINE HEPCIDIN ANTAGONISTS VIFOR (INTERNATIONAL) AG (CH) 2012-08-23 WO disclosed
EP-2200987-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS Boehringer Ingelheim International GmbH (DE) 2010-06-30 EP disclosed
WO-2009030715-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-12 WO disclosed