SCHEMBL3278924

SCHEMBL3278924

CP(=O)(O)ON(c1ccc2cc(-c3ncccn3)ccc2c1)S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.40
F2 P00734 1/20 0.32
KAT6A Q92794 2/20 0.31
ACLY P53396 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2055477 0.80 CYP3A4 (0.41) CYP3A4KAT6A
SCHEMBL2098962 0.78 CYP3A4 (0.38) CYP3A4F2KAT6A
SCHEMBL2055363 0.76 CYP3A4 (0.38) CYP3A4F2
SCHEMBL1319419 0.74 KEAP1 (0.43) CYP3A4
SCHEMBL12115634 0.74 CYP3A4 (0.38) CYP3A4
SCHEMBL3694345 0.73 ALDH1A1 (0.47) CYP3A4
SCHEMBL1110198 0.70 CYP3A4 (0.36) CYP3A4ACLY
SCHEMBL3277272 0.70 ALDH1A1 (0.32) ACLY
SCHEMBL2055412 0.68 CYP3A4 (0.78) CYP3A4ACLY
SCHEMBL3278163 0.67 HCRTR1 (0.38) CYP3A4KAT6AACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2200987-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS Boehringer Ingelheim International GmbH (DE) 2010-06-30 EP disclosed
WO-2009030715-A1 ARYLSULFONYLAMINOMETHYLPHOSPHONIC ACID DERIVATIVES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-12 WO disclosed