SCHEMBL328352

SCHEMBL328352

Nc1ccc2c(c1)N(CCCCl)C(=O)CO2

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.50
POLB P06746 3/20 0.47
TP53 P04637 1/20 0.44
REN P00797 1/20 0.44
HTT P42858 2/20 0.43
TSHR P16473 1/20 0.43
THRB P10828 1/20 0.41
USP2 O75604 1/20 0.41
DRD2 P14416 2/20 0.41
HTR2A P28223 2/20 0.41
MCHR1 Q99705 2/20 0.41
PLK1 P53350 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13071332 0.89 CHRM1 (0.43) KMOPOLBTSHRDRD2HTR2A
SCHEMBL8266002 0.85 POLB (0.49) KMOPOLBTP53RENHTT
SCHEMBL8265502 0.85 POLB (0.49) KMOPOLBTP53RENHTT
SCHEMBL8265365 0.84 POLB (0.56) KMOPOLBTP53HTTTSHR
SCHEMBL4096802 0.84 KMO (0.50) KMOPOLBTP53HTTTSHR
SCHEMBL4102493 0.84 TSHR (0.62) POLBTP53HTTTSHRTHRB
SCHEMBL8879021 0.83 HTT (0.54) KMOPOLBTP53RENHTT
SCHEMBL5799186 0.83 KMO (0.52) KMOPOLBTP53HTTTSHR
SCHEMBL55503 0.83 REN (0.61) KMOPOLBTP53RENHTT
SCHEMBL8264865 0.82 REN (0.57) KMOPOLBTP53RENHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2428508-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND Astellas Pharma Inc. (JP) 2012-03-14 EP disclosed