SCHEMBL3284565

SCHEMBL3284565

COC(=O)c1ccc(-c2ccc(CC3CCN(N4CCC(O[Si](C(C)C)(C(C)C)C(C)C)CC4)C3=O)c(Cl)c2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.35
CHKA P35790 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CMA1 P23946 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PSD A5PKW4 1/20 0.33
MAPT P10636 2/20 0.32
TP53 P04637 1/20 0.32
RHEB Q15382 1/20 0.32
PTGES O14684 1/20 0.32
CHRM4 P08173 2/20 0.31
CHRM2 P08172 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1093032 1.00 ROCK2 (0.35) ROCK2CHKAALDH1A1L3MBTL1CMA1
SCHEMBL1092227 0.92 ROCK2 (0.35) ROCK2CMA1PDE4APDE4BPDE4C
SCHEMBL1094079 0.92 ROCK2 (0.35) ROCK2CMA1PDE4APDE4BPDE4C
SCHEMBL1092143 0.91 CHKA (0.34) CHKAALDH1A1L3MBTL1PDE4APDE4B
SCHEMBL1092145 0.91 CHKA (0.34) CHKAALDH1A1L3MBTL1PDE4APDE4B
SCHEMBL1091733 0.87 LRRK2 (0.35) ROCK2PDE4APDE4BPDE4CPDE4D
SCHEMBL1091734 0.87 LRRK2 (0.35) ROCK2PDE4APDE4BPDE4CPDE4D
SCHEMBL4345635 0.85 P2RX3 (0.34) ROCK2ALDH1A1CHRM2MEN1KMT2A
SCHEMBL1092636 0.83 ROCK2 (0.33) ROCK2
SCHEMBL1092633 0.83 ROCK2 (0.33) ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2021336-B1 INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 LILLY CO ELI (US) 2010-06-30 EP disclosed