SCHEMBL3284835

SCHEMBL3284835

Cc1cn2c(Nc3cc(C)[nH]n3)nc(-c3cc(CNC=O)ccc3F)cc2n1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PLK4 O00444 9/20 0.40
NTRK1 P04629 9/20 0.40
PAK4 O96013 2/20 0.34
RET P07949 5/20 0.34
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
NTRK3 Q16288 1/20 0.33
NTRK2 Q16620 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3288306 0.87 PLK4 (0.40) PLK4NTRK1PAK4RETAURKA
SCHEMBL3045180 0.84 RET (0.49) PLK4NTRK1RETAURKAAURKB
SCHEMBL5262600 0.76 GSK3A (0.41) PLK4NTRK1PAK4RETAURKA
SCHEMBL13221325 0.74 GSK3B (0.54) AURKAAURKB
SCHEMBL3041422 0.73 KDM4E (0.48) NTRK1AURKAAURKB
SCHEMBL15651438 0.72 FGFR4 (0.36) PLK4PAK4AURKAAURKB
SCHEMBL3041030 0.72 GSK3A (0.33) NTRK1RETAURKAAURKB
SCHEMBL3288291 0.72 MAP4K2 (0.41) PLK4PAK4RETAURKAAURKB
SCHEMBL3033835 0.72 RET (0.47) PLK4NTRK1RETAURKAAURKB
SCHEMBL3038694 0.72 GSK3B (0.39) AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7713973-B2 Kinase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-11 US disclosed